Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50042595
TargetSodium-dependent dopamine transporter(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50428288(CHEMBL2338351)
Affinity DataIC50: 290nMAssay Description:Inhibition of human dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50344732(2-chloro-5-(3,5-dioxo-4,5-dihydro-1,2,4-triazin-2(...)
Affinity DataIC50: 800nMAssay Description:Antagonist activity at human P2X7 receptor assessed as inhibition of IL1beta releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50344732(2-chloro-5-(3,5-dioxo-4,5-dihydro-1,2,4-triazin-2(...)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at human P2X7 receptor assessed as inhibition of YOPRO1 accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed