Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50034533
TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50312718(torcetrapib | CHEMBL479527)
Affinity DataIC50: 13nMAssay Description:Inhibition of CETP-mediated BODIPY-labeled cholesteryl ester transfer after 45 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50348222(CHEMBL1800801)
Affinity DataIC50: 93nMAssay Description:Inhibition of CETP-mediated BODIPY-labeled cholesteryl ester transfer after 45 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50331754(methyl 3,5-bis(trifluoromethyl)benzyl((5'-isopropy...)
Affinity DataIC50: 126nMAssay Description:Inhibition of CETP-mediated BODIPY-labeled cholesteryl ester transfer after 45 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50348222(CHEMBL1800801)
Affinity DataIC50: 133nMAssay Description:Inhibition of CETP-mediated BODIPY-labeled cholesteryl ester transfer after 45 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50363940(CHEMBL1951593)
Affinity DataIC50: 293nMAssay Description:Inhibition of CETP-mediated BODIPY-labeled cholesteryl ester transfer after 45 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50363938(CHEMBL1951589)
Affinity DataIC50: 1.42E+4nMAssay Description:Inhibition of CETP-mediated BODIPY-labeled cholesteryl ester transfer after 45 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50363941(CHEMBL1951594)
Affinity DataIC50: 2.73E+4nMAssay Description:Inhibition of CETP-mediated BODIPY-labeled cholesteryl ester transfer after 45 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50363939(CHEMBL1951592)
Affinity DataIC50: 3.72E+4nMAssay Description:Inhibition of CETP-mediated BODIPY-labeled cholesteryl ester transfer after 45 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed