Compile Data Set for Download or QSAR
Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50032960
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336931(N-(3-(4-cyano-3-fluorophenyl)-1-isopropyl-1H-indol...)
Affinity DataIC50: 2.29nMAssay Description:Antagonist activity at human progesterone receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by GRE-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336933(N-(3-(4-cyano-3-methylphenyl)-1-isopropyl-1H-indol...)
Affinity DataIC50: 3.38nMAssay Description:Antagonist activity at human progesterone receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by GRE-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336930((S)-N-(1-sec-butyl-3-(4-cyanophenyl)-1H-indol-6-yl...)
Affinity DataIC50: 3.89nMAssay Description:Antagonist activity at human progesterone receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by GRE-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336934(N-(3-(4-cyanophenyl)-1-isopropyl-1H-indol-6-yl)met...)
Affinity DataIC50: 6.81nMAssay Description:Antagonist activity at human progesterone receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by GRE-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336932(N-(3-(4-cyano-3-methoxyphenyl)-1-isopropyl-1H-indo...)
Affinity DataIC50: 7.28nMAssay Description:Antagonist activity at human progesterone receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by GRE-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336929((R)-N-(1-sec-butyl-3-(4-cyanophenyl)-1H-indol-6-yl...)
Affinity DataIC50: 9.92nMAssay Description:Antagonist activity at human progesterone receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by GRE-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336935(N-(3-(4-cyanophenyl)-1-ethyl-1H-indol-6-yl)methane...)
Affinity DataIC50: 12.6nMAssay Description:Antagonist activity at human progesterone receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by GRE-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50228078((S)-N-(3-(1-cyclopropyl-1-(2,4-difluorophenyl)ethy...)
Affinity DataIC50: 27.2nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50228079((R)-N-(3-(1-cyclopropyl-1-(4-fluorophenyl)ethyl)-1...)
Affinity DataIC50: 64.1nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50228076((R)-N-(3-(1-cyclopropyl-1-(2,4-difluorophenyl)ethy...)
Affinity DataIC50: 306nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336936(N-(3-(4-cyanophenyl)-1-methyl-1H-indol-6-yl)methan...)
Affinity DataIC50: 485nMAssay Description:Antagonist activity at human progesterone receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by GRE-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50228078((S)-N-(3-(1-cyclopropyl-1-(2,4-difluorophenyl)ethy...)
Affinity DataIC50: 715nMAssay Description:Antagonist activity at human progesterone receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by GRE-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50228079((R)-N-(3-(1-cyclopropyl-1-(4-fluorophenyl)ethyl)-1...)
Affinity DataIC50: 765nMAssay Description:Antagonist activity at human progesterone receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by GRE-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50228076((R)-N-(3-(1-cyclopropyl-1-(2,4-difluorophenyl)ethy...)
Affinity DataIC50: 2.02E+3nMAssay Description:Antagonist activity at human progesterone receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by GRE-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336932(N-(3-(4-cyano-3-methoxyphenyl)-1-isopropyl-1H-indo...)
Affinity DataIC50: 2.42E+3nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336937(3-[(4-methoxyphenyl)phenylmethyl]indole | CHEMBL16...)
Affinity DataIC50: 3.72E+3nMAssay Description:Antagonist activity at human progesterone receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by GRE-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336931(N-(3-(4-cyano-3-fluorophenyl)-1-isopropyl-1H-indol...)
Affinity DataIC50: 8.15E+3nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336930((S)-N-(1-sec-butyl-3-(4-cyanophenyl)-1H-indol-6-yl...)
Affinity DataIC50: 9.80E+3nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336929((R)-N-(1-sec-butyl-3-(4-cyanophenyl)-1H-indol-6-yl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336936(N-(3-(4-cyanophenyl)-1-methyl-1H-indol-6-yl)methan...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336935(N-(3-(4-cyanophenyl)-1-ethyl-1H-indol-6-yl)methane...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336934(N-(3-(4-cyanophenyl)-1-isopropyl-1H-indol-6-yl)met...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336933(N-(3-(4-cyano-3-methylphenyl)-1-isopropyl-1H-indol...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336937(3-[(4-methoxyphenyl)phenylmethyl]indole | CHEMBL16...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336931(N-(3-(4-cyano-3-fluorophenyl)-1-isopropyl-1H-indol...)
Affinity DataKi:  0.214nMAssay Description:Displacement of [3H]methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336933(N-(3-(4-cyano-3-methylphenyl)-1-isopropyl-1H-indol...)
Affinity DataKi:  0.298nMAssay Description:Displacement of [3H]methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50228078((S)-N-(3-(1-cyclopropyl-1-(2,4-difluorophenyl)ethy...)
Affinity DataKi:  0.319nMAssay Description:Displacement of [3H]methyltrienolone from human mineralocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336930((S)-N-(1-sec-butyl-3-(4-cyanophenyl)-1H-indol-6-yl...)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50228079((R)-N-(3-(1-cyclopropyl-1-(4-fluorophenyl)ethyl)-1...)
Affinity DataKi:  0.640nMAssay Description:Displacement of [3H]methyltrienolone from human mineralocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336934(N-(3-(4-cyanophenyl)-1-isopropyl-1H-indol-6-yl)met...)
Affinity DataKi:  0.795nMAssay Description:Displacement of [3H]methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336929((R)-N-(1-sec-butyl-3-(4-cyanophenyl)-1H-indol-6-yl...)
Affinity DataKi:  0.834nMAssay Description:Displacement of [3H]methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336932(N-(3-(4-cyano-3-methoxyphenyl)-1-isopropyl-1H-indo...)
Affinity DataKi:  1.45nMAssay Description:Displacement of [3H]methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50228076((R)-N-(3-(1-cyclopropyl-1-(2,4-difluorophenyl)ethy...)
Affinity DataKi:  1.51nMAssay Description:Displacement of [3H]methyltrienolone from human mineralocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336935(N-(3-(4-cyanophenyl)-1-ethyl-1H-indol-6-yl)methane...)
Affinity DataKi:  4.23nMAssay Description:Displacement of [3H]methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50228078((S)-N-(3-(1-cyclopropyl-1-(2,4-difluorophenyl)ethy...)
Affinity DataKi:  5.93nMAssay Description:Displacement of [3H]methyltrienolone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50228079((R)-N-(3-(1-cyclopropyl-1-(4-fluorophenyl)ethyl)-1...)
Affinity DataKi:  6.39nMAssay Description:Displacement of [3H]methyltrienolone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336936(N-(3-(4-cyanophenyl)-1-methyl-1H-indol-6-yl)methan...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336937(3-[(4-methoxyphenyl)phenylmethyl]indole | CHEMBL16...)
Affinity DataKi:  50.2nMAssay Description:Displacement of [3H]methyltrienolone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50228076((R)-N-(3-(1-cyclopropyl-1-(2,4-difluorophenyl)ethy...)
Affinity DataKi:  54.4nMAssay Description:Displacement of [3H]methyltrienolone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336937(3-[(4-methoxyphenyl)phenylmethyl]indole | CHEMBL16...)
Affinity DataKi:  68.9nMAssay Description:Displacement of [3H]methyltrienolone from human androgen receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336937(3-[(4-methoxyphenyl)phenylmethyl]indole | CHEMBL16...)
Affinity DataKi:  86.8nMAssay Description:Displacement of [3H]methyltrienolone from human mineralocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336933(N-(3-(4-cyano-3-methylphenyl)-1-isopropyl-1H-indol...)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]methyltrienolone from human mineralocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336933(N-(3-(4-cyano-3-methylphenyl)-1-isopropyl-1H-indol...)
Affinity DataKi:  157nMAssay Description:Displacement of [3H]methyltrienolone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50228078((S)-N-(3-(1-cyclopropyl-1-(2,4-difluorophenyl)ethy...)
Affinity DataKi:  211nMAssay Description:Displacement of [3H]methyltrienolone from human androgen receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50228079((R)-N-(3-(1-cyclopropyl-1-(4-fluorophenyl)ethyl)-1...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]methyltrienolone from human androgen receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336933(N-(3-(4-cyano-3-methylphenyl)-1-isopropyl-1H-indol...)
Affinity DataKi:  403nMAssay Description:Displacement of [3H]methyltrienolone from human androgen receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50228079((R)-N-(3-(1-cyclopropyl-1-(4-fluorophenyl)ethyl)-1...)
Affinity DataKi:  454nMAssay Description:Displacement of [3H]methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50228078((S)-N-(3-(1-cyclopropyl-1-(2,4-difluorophenyl)ethy...)
Affinity DataKi:  464nMAssay Description:Displacement of [3H]methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336937(3-[(4-methoxyphenyl)phenylmethyl]indole | CHEMBL16...)
Affinity DataKi:  478nMAssay Description:Displacement of [3H]methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336932(N-(3-(4-cyano-3-methoxyphenyl)-1-isopropyl-1H-indo...)
Affinity DataKi:  490nMAssay Description:Displacement of [3H]methyltrienolone from human androgen receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
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