Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50040333
LigandPNGBDBM50392769(CHEMBL2151147)
Affinity DataIC50: 264nMAssay Description:Antagonist activity at Cav3.3 at -80 mV holding potential by whole cell patch clamp analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50392766(CHEMBL2151144)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3S]MK499 from human ERG in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50338167((R)-2-(4-cyclopropylphenyl)-N-(1-(5-(2,2,2-trifluo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3S]MK499 from human ERG in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50392769(CHEMBL2151147)
Affinity DataIC50: 1.20E+4nMAssay Description:Antagonist activity at Cav3.3 at -100 mV holding potential by whole cell patch clamp analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50392768(CHEMBL2151146)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of [3S]MK499 from human ERG in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50392767(CHEMBL2151145)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of [3S]MK499 from human ERG in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50392769(CHEMBL2151147)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of [3S]MK499 from human ERG in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed