Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 50044360
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 915nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 422nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 21nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: >2.50E+3nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 581nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 75nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 313nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 15nMAssay Description:Binding affinity to human DDR2 by Ambit assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 3.80nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by fluorescence spectroscopyMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 15nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 412nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 15nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 18nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 178nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 428nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 252nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 702nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 63nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 406nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 382nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 385nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 424nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 20nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 93nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 230nMAssay Description:Binding affinity to wild type DDR2 (unknown origin) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 3nMAssay Description:Binding affinity to wild type DDR2 (unknown origin) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 33nMAssay Description:Binding affinity to wild type DDR2 (unknown origin) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 98nMAssay Description:Binding affinity to wild type DDR2 (unknown origin) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 6nMAssay Description:Binding affinity to wild type DDR2 (unknown origin) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 7nMAssay Description:Binding affinity to wild type DDR2 (unknown origin) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: 30nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of wild type DDR2 (unknown origin) preincubated for 30 mins before substrate addition by FRET assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of wild type DDR2 (unknown origin) preincubated for 30 mins before substrate addition by FRET assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of wild type DDR2 (unknown origin) preincubated for 30 mins before substrate addition by FRET assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of wild type DDR2 (unknown origin) preincubated for 30 mins before substrate addition by FRET assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of wild type DDR2 (unknown origin) preincubated for 30 mins before substrate addition by FRET assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of wild type DDR2 (unknown origin) preincubated for 30 mins before substrate addition by FRET assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of wild type DDR2 (unknown origin) preincubated for 30 mins before substrate addition by FRET assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of DDR2 (unknown origin) after 120 mins by radiometric assay in presence of gamma-[33P]-ATPMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of wild type DDR2 (unknown origin) preincubated for 30 mins before substrate addition by FRET assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of wild type DDR2 (unknown origin) preincubated for 30 mins before substrate addition by FRET assayMore data for this Ligand-Target Pair
