Compile Data Set for Download or QSAR
Report error Found 79 Enz. Inhib. hit(s) with all data for entry = 50042588
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428185(CHEMBL2336538)
Affinity DataEC50:  8.20nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in CHO cell membranes assessed as inhibition of forskolin-stimulated cAMP production after 4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428180(CHEMBL2336543)
Affinity DataEC50:  2.5nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in CHO cell membranes assessed as inhibition of forskolin-stimulated cAMP production after 4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428174(CHEMBL2336549)
Affinity DataEC50:  73nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in CHO cell membranes assessed as inhibition of forskolin-stimulated cAMP production after 4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428173(CHEMBL2336528)
Affinity DataEC50:  49nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in CHO cell membranes assessed as inhibition of forskolin-stimulated cAMP production after 4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataEC50:  14nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in CHO cell membranes assessed as inhibition of forskolin-stimulated cAMP production after 4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membranes assessed as increase in forskolin-stimulated cAMP production after 45 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399157(CHEMBL2179724)
Affinity DataEC50:  85nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membranes assessed as increase in forskolin-stimulated cAMP production after 45 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428174(CHEMBL2336549)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428180(CHEMBL2336543)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428185(CHEMBL2336538)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428187(CHEMBL2336536)
Affinity DataKi:  9.5nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428186(CHEMBL2336537)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428183(CHEMBL2336540)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428184(CHEMBL2336539)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428178(CHEMBL2336545)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428179(CHEMBL2336544)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428177(CHEMBL2336546)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428173(CHEMBL2336528)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428188(CHEMBL2336535)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428182(CHEMBL2336541)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428194(CHEMBL2336552)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428190(CHEMBL2336566)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428195(CHEMBL2336573)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428175(CHEMBL2336548)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428181(CHEMBL2336542)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428191(CHEMBL2336565)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428193(CHEMBL2336561)
Affinity DataKi:  73nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428176(CHEMBL2336547)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428185(CHEMBL2336538)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428206(CHEMBL2336567)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428192(CHEMBL2336562)
Affinity DataKi:  102nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428189(CHEMBL2336534)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428201(CHEMBL2336530)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428213(CHEMBL2336556)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428214(CHEMBL2336555)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428196(CHEMBL2336529)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428210(CHEMBL2336559)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428203(CHEMBL2336570)
Affinity DataKi:  166nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428217(CHEMBL2336551)
Affinity DataKi:  166nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428208(CHEMBL2336563)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428216(CHEMBL2336553)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428204(CHEMBL2336569)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428184(CHEMBL2336539)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428199(CHEMBL2336532)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428215(CHEMBL2336554)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428211(CHEMBL2336558)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428209(CHEMBL2336560)
Affinity DataKi:  262nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428212(CHEMBL2336557)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
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