Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50044442
TargetAmine oxidase [flavin-containing] A(Human)
Micurx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017198(CHEBI:83326 | TR-701-FA | TEDIZOLID PHOSPHATE)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human recombinant MAO-A expressed in yeast after 1 hr by luciferin-based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetCytochrome P450 2E1(Human)
Micurx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017203(CHEMBL3287379)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of CYP2E1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Micurx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017196(CHEMBL3286407)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in yeast after 1 hr by luciferin-based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Micurx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116067(Zyvox | (S)-N-((3-(3-fluoro-4-morpholinophenyl)-2-...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in yeast after 1 hr by luciferin-based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Micurx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116067(Zyvox | (S)-N-((3-(3-fluoro-4-morpholinophenyl)-2-...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of MAO-A (unknown origin) using tyramine as substrate after 30 to 60 mins by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Micurx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017203(CHEMBL3287379)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in yeast after 1 hr by luciferin-based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Micurx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017205(CHEMBL3287376)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in yeast after 1 hr by luciferin-based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Micurx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017203(CHEMBL3287379)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of MAO-A (unknown origin) using tyramine as substrate after 30 to 60 mins by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Micurx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017204(CHEMBL3287375)
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of human recombinant MAO-A expressed in yeast after 1 hr by luciferin-based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Micurx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017206(CHEMBL3287377)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of human recombinant MAO-A expressed in yeast after 1 hr by luciferin-based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Micurx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017197(CHEMBL3287374)
Affinity DataIC50: 2.70E+5nMAssay Description:Inhibition of human recombinant MAO-A expressed in yeast after 1 hr by luciferin-based luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed