Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50044099
TargetBifunctional epoxide hydrolase 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM25731(CHEMBL1458 | 1,3-dicyclohexylurea | US8815951, 1,3...)
Affinity DataIC50: 25nMAssay Description:Inhibition of human full-length C-terminal His6-tagged sEH expressed in Escherichia coli BL21(DE3) cells using PHOME as substrate incubated with enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50001939(CHEMBL1873898)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of human full-length C-terminal His6-tagged sEH expressed in Escherichia coli BL21(DE3) cells using PHOME as substrate incubated with enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBifunctional epoxide hydrolase 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50001937(CHEMBL3233603)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of human full-length C-terminal His6-tagged sEH expressed in Escherichia coli BL21(DE3) cells using PHOME as substrate incubated with enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBifunctional epoxide hydrolase 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50001938(CHEMBL3233604)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human full-length C-terminal His6-tagged sEH expressed in Escherichia coli BL21(DE3) cells using PHOME as substrate incubated with enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBifunctional epoxide hydrolase 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50002344(CHEMBL3233607)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of human full-length C-terminal His6-tagged sEH expressed in Escherichia coli BL21(DE3) cells using PHOME as substrate incubated with enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBifunctional epoxide hydrolase 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50002341(CHEMBL442384)
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of human full-length C-terminal His6-tagged sEH expressed in Escherichia coli BL21(DE3) cells using PHOME as substrate incubated with enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBifunctional epoxide hydrolase 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50002348(CHEMBL2094355 | DNDI1416972)
Affinity DataIC50: 6.10E+4nMAssay Description:Inhibition of human full-length C-terminal His6-tagged sEH expressed in Escherichia coli BL21(DE3) cells using PHOME as substrate incubated with enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBifunctional epoxide hydrolase 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50002342(CHEMBL3233606)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of human full-length C-terminal His6-tagged sEH expressed in Escherichia coli BL21(DE3) cells using PHOME as substrate incubated with enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBifunctional epoxide hydrolase 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50001940(CHEMBL3233605)
Affinity DataIC50: 1.27E+5nMAssay Description:Inhibition of human full-length C-terminal His6-tagged sEH expressed in Escherichia coli BL21(DE3) cells using PHOME as substrate incubated with enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBifunctional epoxide hydrolase 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50002352(CHEMBL3233609)
Affinity DataIC50: 1.71E+5nMAssay Description:Inhibition of human full-length C-terminal His6-tagged sEH expressed in Escherichia coli BL21(DE3) cells using PHOME as substrate incubated with enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBifunctional epoxide hydrolase 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50002351(CHEMBL3233608)
Affinity DataIC50: 1.95E+5nMAssay Description:Inhibition of human full-length C-terminal His6-tagged sEH expressed in Escherichia coli BL21(DE3) cells using PHOME as substrate incubated with enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)