Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50044175
TargetHistone deacetylase 6(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007730(CHEMBL3233755)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of human HDAC-6 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007729(CHEMBL3233488)
Affinity DataIC50: 29nMAssay Description:Displacement of GM-FTC from Hsp90-alpha (unknown origin) after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 29nMAssay Description:Inhibition of human HDAC-6 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007730(CHEMBL3233755)
Affinity DataIC50: 33nMAssay Description:Displacement of GM-FTC from Hsp90-alpha (unknown origin) after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007731(CHEMBL3233754)
Affinity DataIC50: 34nMAssay Description:Displacement of GM-FTC from Hsp90-alpha (unknown origin) after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007732(CHEMBL3233752)
Affinity DataIC50: 54nMAssay Description:Displacement of GM-FTC from Hsp90-alpha (unknown origin) after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM20926(5-[2,4-dihydroxy-5-(propan-2-yl)phenyl]-N-ethyl-4-...)
Affinity DataIC50: 61nMAssay Description:Displacement of GM-FTC from Hsp90-alpha (unknown origin) after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007733(CHEMBL3233753)
Affinity DataIC50: 68nMAssay Description:Displacement of GM-FTC from Hsp90-alpha (unknown origin) after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007734(CHEMBL3233485)
Affinity DataIC50: 100nMAssay Description:Displacement of GM-FTC from Hsp90-alpha (unknown origin) after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007735(CHEMBL3233486)
Affinity DataIC50: 110nMAssay Description:Displacement of GM-FTC from Hsp90-alpha (unknown origin) after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007736(CHEMBL3233483)
Affinity DataIC50: 160nMAssay Description:Displacement of GM-FTC from Hsp90-alpha (unknown origin) after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 243nMAssay Description:Inhibition of human HDAC-8 using RHK(Ac)K(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 1(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 258nMAssay Description:Inhibition of human HDAC-1 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 7(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 344nMAssay Description:Inhibition of human HDAC-7 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 350nMAssay Description:Inhibition of human HDAC-3/NCOR-2 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistone deacetylase 11(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 362nMAssay Description:Inhibition of human HDAC-11 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistone deacetylase 5(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 378nMAssay Description:Inhibition of human HDAC-5 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetPolyamine deacetylase HDAC10(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 456nMAssay Description:Inhibition of human HDAC-10 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 493nMAssay Description:Inhibition of human HDAC-4 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistone deacetylase 11(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007730(CHEMBL3233755)
Affinity DataIC50: 521nMAssay Description:Inhibition of human HDAC-11 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetPolyamine deacetylase HDAC10(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007730(CHEMBL3233755)
Affinity DataIC50: 886nMAssay Description:Inhibition of human HDAC-10 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 921nMAssay Description:Inhibition of human HDAC-2 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHeat shock protein HSP 90-alpha(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007737(CHEMBL3233487)
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of GM-FTC from Hsp90-alpha (unknown origin) after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007738(CHEMBL3233750)
Affinity DataIC50: 1.40E+3nMAssay Description:Displacement of GM-FTC from Hsp90-alpha (unknown origin) after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistone deacetylase 5(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007730(CHEMBL3233755)
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of human HDAC-5 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007730(CHEMBL3233755)
Affinity DataIC50: 1.76E+3nMAssay Description:Inhibition of human HDAC-8 using RHK(Ac)K(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007730(CHEMBL3233755)
Affinity DataIC50: 2.03E+3nMAssay Description:Inhibition of human HDAC-1 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistone deacetylase 7(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007730(CHEMBL3233755)
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of human HDAC-7 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007740(CHEMBL3233484)
Affinity DataIC50: 3.90E+3nMAssay Description:Displacement of GM-FTC from Hsp90-alpha (unknown origin) after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
LigandPNGBDBM50007730(CHEMBL3233755)
Affinity DataIC50: 4.23E+3nMAssay Description:Inhibition of human HDAC-3/NCOR-2 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007730(CHEMBL3233755)
Affinity DataIC50: 9.49E+3nMAssay Description:Inhibition of human HDAC-2 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007730(CHEMBL3233755)
Affinity DataIC50: 7.59E+4nMAssay Description:Inhibition of human HDAC-4 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007741(CHEMBL3233482)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of GM-FTC from Hsp90-alpha (unknown origin) after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007742(CHEMBL3233489)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of GM-FTC from Hsp90-alpha (unknown origin) after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50007743(CHEMBL3233490)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of GM-FTC from Hsp90-alpha (unknown origin) after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed