Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50043915
TargetNuclear receptor ROR-alpha(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50448405(CHEMBL3121750)
Affinity DataIC50: 1.30E+3nMAssay Description:Inverse agonist activity at human RORalpha expressed in HEK293 cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50448405(CHEMBL3121750)
Affinity DataIC50: 4.50E+3nMAssay Description:Inverse agonist activity at human RORgamma expressed in HEK293 cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50448404(CHEMBL3121751)
Affinity DataIC50: 1.00E+4nMAssay Description:Inverse agonist activity at human RORgamma expressed in HEK293 cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50448404(CHEMBL3121751)
Affinity DataIC50: 1.00E+4nMAssay Description:Inverse agonist activity at human RORbeta expressed in HEK293 cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50448405(CHEMBL3121750)
Affinity DataIC50: 1.00E+4nMAssay Description:Inverse agonist activity at human RORbeta expressed in HEK293 cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50448404(CHEMBL3121751)
Affinity DataIC50: 1.00E+4nMAssay Description:Inverse agonist activity at human RORalpha expressed in HEK293 cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed