Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50005973
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495835(CHEMBL3113234)
Affinity DataIC50: 90nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495841(CHEMBL3113239)
Affinity DataIC50: 240nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495849(CHEMBL3113224)
Affinity DataIC50: 260nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495840(CHEMBL3113240)
Affinity DataIC50: 270nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495846(CHEMBL3113235)
Affinity DataIC50: 300nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495840(CHEMBL3113240)
Affinity DataIC50: 300nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 350nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495841(CHEMBL3113239)
Affinity DataIC50: 440nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495831(CHEMBL3113231)
Affinity DataIC50: 550nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50056999(CHEMBL56367 | nimesulide)
Affinity DataIC50: 700nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495831(CHEMBL3113231)
Affinity DataIC50: 710nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495833(CHEMBL3113229)
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495832(CHEMBL3113237)
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495839(CHEMBL3113241)
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495835(CHEMBL3113234)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495847(CHEMBL3113233)
Affinity DataIC50: 1.47E+3nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495845(CHEMBL3113236)
Affinity DataIC50: 1.57E+3nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495845(CHEMBL3113236)
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495849(CHEMBL3113224)
Affinity DataIC50: 1.93E+3nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495847(CHEMBL3113233)
Affinity DataIC50: 1.96E+3nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495844(CHEMBL3113242)
Affinity DataIC50: 2.09E+3nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495832(CHEMBL3113237)
Affinity DataIC50: 2.27E+3nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495846(CHEMBL3113235)
Affinity DataIC50: 2.32E+3nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495836(CHEMBL3113232)
Affinity DataIC50: 3.28E+3nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495842(CHEMBL3113228)
Affinity DataIC50: 3.61E+3nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50056999(CHEMBL56367 | nimesulide)
Affinity DataIC50: 3.76E+3nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495833(CHEMBL3113229)
Affinity DataIC50: 4.11E+3nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495834(CHEMBL3113238)
Affinity DataIC50: 4.21E+3nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495843(CHEMBL3113226)
Affinity DataIC50: 6.65E+3nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495839(CHEMBL3113241)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495837(CHEMBL3113230)
Affinity DataIC50: 1.49E+4nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495838(CHEMBL3113225)
Affinity DataIC50: 1.81E+4nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495848(CHEMBL3113227)
Affinity DataIC50: 1.96E+4nMAssay Description:Inhibition of COX-1 in human whole blood assessed as thromboxane B2 level in serum after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495844(CHEMBL3113242)
Affinity DataIC50: 2.07E+4nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495836(CHEMBL3113232)
Affinity DataIC50: 3.07E+4nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495842(CHEMBL3113228)
Affinity DataIC50: 3.51E+4nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495843(CHEMBL3113226)
Affinity DataIC50: 3.62E+4nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495848(CHEMBL3113227)
Affinity DataIC50: 5.68E+4nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495838(CHEMBL3113225)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495837(CHEMBL3113230)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50495834(CHEMBL3113238)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of COX-2 in human whole blood assessed as PGE2 level in plasma after 5 mins by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed