Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50043757
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50220136(CHEMBL1471 | 5-(((2R,3S)-2-((R)-1-(3,5-bis(trifluo...)
Affinity DataKi:  0.0794nMAssay Description:Binding affinity to NK1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50291261(SR-14280 | SR-142801 | (S)-(+)-N-((3-[1-Benzoyl-3-...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to NK3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50051293(SB-2234 | 3-Hydroxy-2-phenyl-quinoline-4-carboxyli...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I][MePhe7]neurokinin B from human NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445808(CHEMBL3104784)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445808(CHEMBL3104784)
Affinity DataKi:  13nMAssay Description:Binding affinity to NK1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445809(CHEMBL3104786)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445808(CHEMBL3104784)
Affinity DataKi:  72nMAssay Description:Binding affinity to NK3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445808(CHEMBL3104784)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445807(CHEMBL3104778)
Affinity DataKi:  79nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445806(CHEMBL3104782)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445805(CHEMBL3104774)
Affinity DataKi:  251nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445804(CHEMBL3104780)
Affinity DataKi:  251nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445803(CHEMBL3104775)
Affinity DataKi:  316nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445802(CHEMBL3104777)
Affinity DataKi:  316nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445818(CHEMBL3104773)
Affinity DataKi:  794nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445806(CHEMBL3104782)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445817(CHEMBL3104776)
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445816(CHEMBL3104781)
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445820(CHEMBL3104783)
Affinity DataKi:  3.98E+3nMAssay Description:Binding affinity to NK3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445819(CHEMBL3104785)
Affinity DataKi:  5.01E+3nMAssay Description:Binding affinity to NK3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445805(CHEMBL3104774)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445803(CHEMBL3104775)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445807(CHEMBL3104778)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445804(CHEMBL3104780)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445809(CHEMBL3104786)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445815(CHEMBL3104769)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445818(CHEMBL3104773)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445817(CHEMBL3104776)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445802(CHEMBL3104777)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445811(CHEMBL3104779)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445816(CHEMBL3104781)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445810(CHEMBL3104768)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445814(CHEMBL3104770)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445813(CHEMBL3104771)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445812(CHEMBL3104772)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445811(CHEMBL3104779)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445815(CHEMBL3104769)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445814(CHEMBL3104770)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445813(CHEMBL3104771)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445812(CHEMBL3104772)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50445810(CHEMBL3104768)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [125I]-Bolton Hunter-Substance P from human NK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed