Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50044061
TargetVascular endothelial growth factor receptor 2(Human)
Comenius University

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataIC50: 13nMAssay Description:Inhibition of GST-tagged recombinant human VEGFR2 expressed in Sf9 cells by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetVascular endothelial growth factor receptor 2(Human)
Comenius University

Curated by ChEMBL
LigandPNGBDBM50005215(CHEMBL3109274)
Affinity DataIC50: 15nMAssay Description:Inhibition of GST-tagged recombinant human VEGFR2 expressed in Sf9 cells by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Comenius University

Curated by ChEMBL
LigandPNGBDBM5875(N-[5-(ethanesulfonyl)-2-methoxyphenyl]-5-[3-(pyrid...)
Affinity DataIC50: 17nMAssay Description:Inhibition of GST-tagged recombinant human VEGFR2 expressed in Sf9 cells by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Comenius University

Curated by ChEMBL
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataIC50: 31nMAssay Description:Inhibition of GST-tagged recombinant human VEGFR2 expressed in Sf9 cells by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Comenius University

Curated by ChEMBL
LigandPNGBDBM50005212(CHEMBL3109275)
Affinity DataIC50: 51nMAssay Description:Inhibition of GST-tagged recombinant human VEGFR2 expressed in Sf9 cells by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Comenius University

Curated by ChEMBL
LigandPNGBDBM50005213(CHEMBL3109276)
Affinity DataIC50: 170nMAssay Description:Inhibition of GST-tagged recombinant human VEGFR2 expressed in Sf9 cells by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Comenius University

Curated by ChEMBL
LigandPNGBDBM50005214(CHEMBL3109277)
Affinity DataIC50: 202nMAssay Description:Inhibition of GST-tagged recombinant human VEGFR2 expressed in Sf9 cells by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMed