Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50043740
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50125099(1-benzyl-4-(4-methoxybenzyl)piperazine | 1-Benzyl-...)
Affinity DataKi:  0.470nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50445477(CHEMBL3104856)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50445476(CHEMBL3104857)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50257493((R)-(1-benzyl-4-(4-methoxybenzyl)piperazin-2-yl)me...)
Affinity DataKi:  12nMAssay Description:Binding affinity to sigma-1 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50048866(1-cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronap...)
Affinity DataKi:  13nMAssay Description:Binding affinity to sigma-1 receptor in human MCF7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50445476(CHEMBL3104857)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in human RPMI8226 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Greifswald

Curated by ChEMBL
LigandPNGBDBM50445477(CHEMBL3104856)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in human RPMI8226 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed