Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50043597
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50382559(ISPINESIB)
Affinity DataIC50: 5nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443437(CHEMBL3087419)
Affinity DataIC50: 23nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443438(CHEMBL3087418)
Affinity DataIC50: 27nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443436(CHEMBL3087420)
Affinity DataIC50: 38nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443425(CHEMBL3087430)
Affinity DataIC50: 52nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443426(CHEMBL3087429)
Affinity DataIC50: 59nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443427(CHEMBL3087428)
Affinity DataIC50: 63nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443429(CHEMBL3087426)
Affinity DataIC50: 67nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443430(CHEMBL3087425)
Affinity DataIC50: 76nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443428(CHEMBL3087427)
Affinity DataIC50: 78nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443435(CHEMBL3087421)
Affinity DataIC50: 91nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443439(CHEMBL3087417)
Affinity DataIC50: 98nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443441(CHEMBL3087415)
Affinity DataIC50: 122nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443440(CHEMBL3087416)
Affinity DataIC50: 123nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443442(CHEMBL3087414)
Affinity DataIC50: 134nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443431(CHEMBL3087424)
Affinity DataIC50: 149nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443432(CHEMBL3087423)
Affinity DataIC50: 157nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443434(CHEMBL3087422)
Affinity DataIC50: 168nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50443433(CHEMBL3085794)
Affinity DataIC50: 170nMAssay Description:Inhibition of C-terminal His-tagged microtubule-stimulated KSP motor domain (1 to 369) ATPase activity (unknown origin) preincubated for 30 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed