Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50005780
TargetCannabinoid receptor 2(Human)
National Institute On Aging

Curated by ChEMBL
LigandPNGBDBM50494417(CHEMBL3086844)
Affinity DataEC50:  42nMAssay Description:Agonist activity at CB2 receptor (unknown origin) after 90 to 180 mins by beta-arrestin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
National Institute On Aging

Curated by ChEMBL
LigandPNGBDBM50494419(Tetrahydrobungeanool)
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells preincubated for 1 hr followed by radioligand addition measured after 1 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Aging

Curated by ChEMBL
LigandPNGBDBM50494416(Hydroxy-Beta-Sanshool | CHEMBL2335715)
Affinity DataIC50: 9nMAssay Description:Displacement of [3H]-Win55212-2 from human CB1 receptor expressed in CHO cells preincubated for 1 hr followed by radioligand addition measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Aging

Curated by ChEMBL
LigandPNGBDBM50494422(CHEMBL3086847)
Affinity DataIC50: 41nMAssay Description:Displacement of [3H]-Win55212-2 from human CB1 receptor expressed in CHO cells preincubated for 1 hr followed by radioligand addition measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
National Institute On Aging

Curated by ChEMBL
LigandPNGBDBM50318477(Hydroxy-alpha-sanshool | CHEMBL1084610)
Affinity DataIC50: 59nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells preincubated for 1 hr followed by radioligand addition measured after 1 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Aging

Curated by ChEMBL
LigandPNGBDBM50494417(CHEMBL3086844)
Affinity DataIC50: 100nMAssay Description:Displacement of [3H]-Win55212-2 from human CB1 receptor expressed in CHO cells preincubated for 1 hr followed by radioligand addition measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
National Institute On Aging

Curated by ChEMBL
LigandPNGBDBM50494416(Hydroxy-Beta-Sanshool | CHEMBL2335715)
Affinity DataIC50: 131nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells preincubated for 1 hr followed by radioligand addition measured after 1 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
National Institute On Aging

Curated by ChEMBL
LigandPNGBDBM50494422(CHEMBL3086847)
Affinity DataIC50: 168nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells preincubated for 1 hr followed by radioligand addition measured after 1 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Aging

Curated by ChEMBL
LigandPNGBDBM50494421(CHEBI:81359 | CHEMBL3086846)
Affinity DataIC50: 184nMAssay Description:Displacement of [3H]-Win55212-2 from human CB1 receptor expressed in CHO cells preincubated for 1 hr followed by radioligand addition measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
National Institute On Aging

Curated by ChEMBL
LigandPNGBDBM50494421(CHEBI:81359 | CHEMBL3086846)
Affinity DataIC50: 197nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells preincubated for 1 hr followed by radioligand addition measured after 1 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
National Institute On Aging

Curated by ChEMBL
LigandPNGBDBM50494420(CHEMBL3086845)
Affinity DataIC50: 224nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells preincubated for 1 hr followed by radioligand addition measured after 1 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
National Institute On Aging

Curated by ChEMBL
LigandPNGBDBM50494417(CHEMBL3086844)
Affinity DataIC50: 664nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells preincubated for 1 hr followed by radioligand addition measured after 1 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Aging

Curated by ChEMBL
LigandPNGBDBM50494420(CHEMBL3086845)
Affinity DataIC50: 1.39E+3nMAssay Description:Displacement of [3H]-Win55212-2 from human CB1 receptor expressed in CHO cells preincubated for 1 hr followed by radioligand addition measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Aging

Curated by ChEMBL
LigandPNGBDBM50494418(CHEMBL505802)
Affinity DataIC50: 2.40E+3nMAssay Description:Displacement of [3H]-Win55212-2 from human CB1 receptor expressed in CHO cells preincubated for 1 hr followed by radioligand addition measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Aging

Curated by ChEMBL
LigandPNGBDBM50494419(Tetrahydrobungeanool)
Affinity DataIC50: 4.60E+3nMAssay Description:Displacement of [3H]-Win55212-2 from human CB1 receptor expressed in CHO cells preincubated for 1 hr followed by radioligand addition measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Aging

Curated by ChEMBL
LigandPNGBDBM50318477(Hydroxy-alpha-sanshool | CHEMBL1084610)
Affinity DataIC50: 7.40E+3nMAssay Description:Displacement of [3H]-Win55212-2 from human CB1 receptor expressed in CHO cells preincubated for 1 hr followed by radioligand addition measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
National Institute On Aging

Curated by ChEMBL
LigandPNGBDBM50494418(CHEMBL505802)
Affinity DataIC50: 9.10E+3nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells preincubated for 1 hr followed by radioligand addition measured after 1 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed