Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50005908
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM13533(1-[5-tert-butyl-2-(p-tolyl)pyrazol-3-yl]-3-[4-(2-m...)
Affinity DataIC50: 8nMAssay Description:Inhibition of human p38-MAPKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50495335(CHEMBL3109731)
Affinity DataIC50: 65nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50495336(CHEMBL3109732)
Affinity DataIC50: 196nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM13345(3-(3-tert-butyl-1H-pyrazol-5-yl)-1-{4-chloro-3-[(p...)
Affinity DataIC50: 350nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM13337(3-(benzyloxy)pyridin-2-amine | Pyridine derived fr...)
Affinity DataIC50: 1.30E+6nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)