Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50001491
TargetThromboxane A2 receptor(Human)
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50015847(CHEMBL312732 | 7-(3-{[2-(5-Cyclohexyl-pentanoylami...)
Affinity DataKd:  2.60nMAssay Description:Binding affinity was determined from the inhibition of [3H]-SQ 29,548 binding to Thromboxane A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50015848(CHEMBL79287 | 7-{3-[(2-Heptanethioylamino-acetylam...)
Affinity DataKd:  12nMAssay Description:Binding affinity was determined from the inhibition of [3H]-SQ 29,548 binding to Thromboxane A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50015849(CHEMBL81263 | 7-{3-[(2-Octanoylamino-acetylamino)-...)
Affinity DataKd:  50nMAssay Description:Binding affinity was determined from the inhibition of [3H]-SQ 29,548 binding to Thromboxane A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50015850(CHEMBL79278 | 7-(3-{[2-(2-Phenylsulfanyl-acetylami...)
Affinity DataKd:  41nMAssay Description:Binding affinity was determined from the inhibition of [3H]-SQ 29,548 binding to Thromboxane A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50015852(CHEMBL82146 | 7-{3-[(2-Nonanoylamino-acetylamino)-...)
Affinity DataKd:  8.30nMAssay Description:Binding affinity was determined from the inhibition of [3H]-SQ 29,548 binding to Thromboxane A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50015851(CHEMBL83366 | 7-[3-({2-[2-(4-tert-Butyl-phenylsulf...)
Affinity DataKd:  4.20nMAssay Description:Binding affinity was determined from the inhibition of [3H]-SQ 29,548 binding to Thromboxane A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50015853(CHEMBL310406 | 7-(3-{[2-(4-Cyclohexyl-butyrylamino...)
Affinity DataKd:  1.10nMAssay Description:Binding affinity was determined from the inhibition of [3H]-SQ 29,548 binding to Thromboxane A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50015854(CHEMBL312360 | 7-{3-[(2-Heptanethioylamino-thioace...)
Affinity DataKd:  26nMAssay Description:Binding affinity was determined from the inhibition of [3H]-SQ 29,548 binding to Thromboxane A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50015849(CHEMBL81263 | 7-{3-[(2-Octanoylamino-acetylamino)-...)
Affinity DataKd:  49.6nMAssay Description:Binding affinity was determined from the inhibition of [3H]-SQ 29,548 binding to Thromboxane A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed