Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50005596
TargetSodium channel protein type 2 subunit alpha(Human)
Institute of Nuclear Medicine

Curated by ChEMBL
LigandPNGBDBM50493060(CHEMBL2419774)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human voltage-gated sodium channel subunit alpha Nav1.2 expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Institute of Nuclear Medicine

Curated by ChEMBL
LigandPNGBDBM50030510([1-Benzyl-7-chloro-1H-quinolin-(4E)-ylidene]-penty...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human voltage-gated sodium channel subunit alpha Nav1.2 expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Institute of Nuclear Medicine

Curated by ChEMBL
LigandPNGBDBM50030510([1-Benzyl-7-chloro-1H-quinolin-(4E)-ylidene]-penty...)
Affinity DataKi:  9nMAssay Description:Inhibition of rat brain voltage-gated sodium channel subunit alpha Nav1.2-mediated current expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed