Compile Data Set for Download or QSAR
Report error Found 124 Enz. Inhib. hit(s) with all data for entry = 50043168
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436963(CHEMBL2402255)
Affinity DataIC50: 6.30nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436963(CHEMBL2402255)
Affinity DataIC50: 9.5nMAssay Description:Antagonist activity at P2Y12 receptor in human washed platelets assessed as inhibition of fibrinogen-induced aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436962(CHEMBL2402264)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at P2Y12 receptor in human washed platelets assessed as inhibition of fibrinogen-induced aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436961(CHEMBL2402266)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at P2Y12 receptor in human washed platelets assessed as inhibition of fibrinogen-induced aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436963(CHEMBL2402255)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436960(CHEMBL2402260)
Affinity DataIC50: 26nMAssay Description:Antagonist activity at P2Y12 receptor in human washed platelets assessed as inhibition of fibrinogen-induced aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436960(CHEMBL2402260)
Affinity DataIC50: 27nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436958(CHEMBL2402144)
Affinity DataIC50: 31nMAssay Description:Antagonist activity at P2Y12 receptor in human washed platelets assessed as inhibition of fibrinogen-induced aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436952(CHEMBL2402142)
Affinity DataIC50: 31nMAssay Description:Antagonist activity at P2Y12 receptor in human washed platelets assessed as inhibition of fibrinogen-induced aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436961(CHEMBL2402266)
Affinity DataIC50: 33nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436962(CHEMBL2402264)
Affinity DataIC50: 34nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436958(CHEMBL2402144)
Affinity DataIC50: 37nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436957(CHEMBL2402244)
Affinity DataIC50: 38nMAssay Description:Antagonist activity at P2Y12 receptor in human washed platelets assessed as inhibition of fibrinogen-induced aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436957(CHEMBL2402244)
Affinity DataIC50: 39nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436962(CHEMBL2402264)
Affinity DataIC50: 42nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436961(CHEMBL2402266)
Affinity DataIC50: 54nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436960(CHEMBL2402260)
Affinity DataIC50: 57nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436959(CHEMBL2402257)
Affinity DataIC50: 62nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436958(CHEMBL2402144)
Affinity DataIC50: 64nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436934(CHEMBL2402249)
Affinity DataIC50: 68nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436953(CHEMBL2402258)
Affinity DataIC50: 78nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436949(CHEMBL2402259)
Affinity DataIC50: 79nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436957(CHEMBL2402244)
Affinity DataIC50: 79nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436949(CHEMBL2402259)
Affinity DataIC50: 82nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436953(CHEMBL2402258)
Affinity DataIC50: 86nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436956(CHEMBL2402263)
Affinity DataIC50: 88nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436954(CHEMBL2402248)
Affinity DataIC50: 90nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436955(CHEMBL2402251)
Affinity DataIC50: 90nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436953(CHEMBL2402258)
Affinity DataIC50: 94nMAssay Description:Antagonist activity at P2Y12 receptor in human washed platelets assessed as inhibition of fibrinogen-induced aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436951(CHEMBL2402149)
Affinity DataIC50: 95nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436952(CHEMBL2402142)
Affinity DataIC50: 95nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436934(CHEMBL2402249)
Affinity DataIC50: 97nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436955(CHEMBL2402251)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436971(CHEMBL2402151)
Affinity DataIC50: 110nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436952(CHEMBL2402142)
Affinity DataIC50: 110nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50345265(Ethyl 5-cyano-6-(4-{[(4-fluorobenzyl)amino]carbony...)
Affinity DataIC50: 110nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436970(CHEMBL2402245)
Affinity DataIC50: 120nMAssay Description:Antagonist activity at P2Y12 receptor in human washed platelets assessed as inhibition of fibrinogen-induced aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436954(CHEMBL2402248)
Affinity DataIC50: 120nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436972(CHEMBL2402265)
Affinity DataIC50: 130nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436971(CHEMBL2402151)
Affinity DataIC50: 140nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436972(CHEMBL2402265)
Affinity DataIC50: 140nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436951(CHEMBL2402149)
Affinity DataIC50: 150nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436956(CHEMBL2402263)
Affinity DataIC50: 150nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436967(CHEMBL2402272)
Affinity DataIC50: 150nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436954(CHEMBL2402248)
Affinity DataIC50: 160nMAssay Description:Antagonist activity at P2Y12 receptor in human washed platelets assessed as inhibition of fibrinogen-induced aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436970(CHEMBL2402245)
Affinity DataIC50: 170nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436931(CHEMBL2402267)
Affinity DataIC50: 180nMAssay Description:Displacement of [125I]-AZ11931285 from P2Y12 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436959(CHEMBL2402257)
Affinity DataIC50: 190nMAssay Description:Antagonist activity at P2Y12 receptor in human washed platelets assessed as inhibition of fibrinogen-induced aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436965(CHEMBL2402273)
Affinity DataIC50: 190nMAssay Description:Antagonist activity at P2Y12 receptor in human washed platelets assessed as inhibition of fibrinogen-induced aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50436959(CHEMBL2402257)
Affinity DataIC50: 190nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) assessed as inhibition of GTPgammaS binding after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Displayed 1 to 50 (of 124 total ) | Next | Last >>
Jump to: