Compile Data Set for Download or QSAR
Report error Found 193 Enz. Inhib. hit(s) with all data for entry = 50035891
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50009552(CHA | CHEMBL45891 | N6-Cyclohexylado (CHA) | 2-[6-...)
Affinity DataIC50: 2nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50009552(CHA | CHEMBL45891 | N6-Cyclohexylado (CHA) | 2-[6-...)
Affinity DataIC50: 2nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50118810(CHEMBL139000 | N6-[(R)-1-Methyl-2-phenylethyl]ado ...)
Affinity DataIC50: 2.40nMAssay Description:Evaluated for the binding affinity towards the Adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004566(CHEMBL268431 | 9-chloro-2-(furan-2-yl)-[1,2,4]tria...)
Affinity DataIC50: 2.80nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004584(CHEMBL72669 | (8-Chloro-1-trifluoromethyl-[1,2,4]t...)
Affinity DataIC50: 5.5nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004566(CHEMBL268431 | 9-chloro-2-(furan-2-yl)-[1,2,4]tria...)
Affinity DataIC50: 6nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM42467(N6-PHENYLADENOSINE | cid_101430 | (2R,3R,4S,5R)-2-...)
Affinity DataIC50: 6.5nMAssay Description:Evaluated for the binding affinity towards the Adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataIC50: 10nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataIC50: 17nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015751(CHEMBL72517 | (8-Chloro-1-ethyl-[1,2,4]triazolo[4,...)
Affinity DataIC50: 20nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004571(CHEMBL303198 | CP-66713 | 8-Chloro-1-phenyl-[1,2,4...)
Affinity DataIC50: 21nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015779(CHEMBL312449 | 7,8-Dichloro-1-ethyl-[1,2,4]triazol...)
Affinity DataIC50: 23nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015773(CHEMBL311616 | (8-Chloro-1-trifluoromethyl-[1,2,4]...)
Affinity DataIC50: 24nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015801(CHEMBL420368 | (8-Chloro-1-pentafluoroethyl-[1,2,4...)
Affinity DataIC50: 24nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015765(CHEMBL72051 | 8-Chloro-1-ethyl-[1,2,4]triazolo[4,3...)
Affinity DataIC50: 28nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015803(CHEMBL73478 | (8-Chloro-1-trifluoromethyl-[1,2,4]t...)
Affinity DataIC50: 28nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015810(CHEMBL73181 | 7-Chloro-1-ethyl-[1,2,4]triazolo[4,3...)
Affinity DataIC50: 29nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015770(CHEMBL306351 | Cyclohexyl-(8-fluoro-1-trifluoromet...)
Affinity DataIC50: 32nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015829(CHEMBL73095 | 8-Chloro-1-(4-chloro-phenyl)-[1,2,4]...)
Affinity DataIC50: 33nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015784(CHEMBL431376 | 1-Ethyl-7-methoxy-[1,2,4]triazolo[4...)
Affinity DataIC50: 36nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015798(CHEMBL307187 | 8-Chloro-1-trifluoromethyl-[1,2,4]t...)
Affinity DataIC50: 44nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015794(CHEMBL73747 | (8-Chloro-1-ethyl-[1,2,4]triazolo[4,...)
Affinity DataIC50: 44nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015817(CHEMBL442176 | (8-Fluoro-1-trifluoromethyl-[1,2,4]...)
Affinity DataIC50: 57nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015752(CHEMBL72177 | (8-Chloro-1-ethyl-[1,2,4]triazolo[4,...)
Affinity DataIC50: 60nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015771(CHEMBL72052 | 1-Ethyl-[1,2,4]triazolo[4,3-a]quinox...)
Affinity DataIC50: 62nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015798(CHEMBL307187 | 8-Chloro-1-trifluoromethyl-[1,2,4]t...)
Affinity DataIC50: 65nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015810(CHEMBL73181 | 7-Chloro-1-ethyl-[1,2,4]triazolo[4,3...)
Affinity DataIC50: 75nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM15336(1-methyl-3-(2-methylpropyl)-2,3,6,7-tetrahydro-1H-...)
Affinity DataIC50: 100nMAssay Description:Evaluated for Ca++ dependent phosphodiesterase activity. More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015788(CHEMBL312744 | 7-Methoxy-[1,2,4]triazolo[4,3-a]qui...)
Affinity DataIC50: 100nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50015800(CHEMBL310041 | Diethyl-(1-ethyl-[1,2,4]triazolo[4,...)
Affinity DataIC50: 100nMAssay Description:Evaluated for Ca++ dependent phosphodiesterase activity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015748(CHEMBL311481 | 8-Fluoro-1-trifluoromethyl-[1,2,4]t...)
Affinity DataIC50: 100nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015806(CHEMBL70435 | (8-Chloro-1-methyl-[1,2,4]triazolo[4...)
Affinity DataIC50: 100nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080398(N6-[(S)-1-Methyl-2-phenylethyl]ado (S-PIA) | CHEMB...)
Affinity DataIC50: 105nMAssay Description:Evaluated for the binding affinity towards the Adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015765(CHEMBL72051 | 8-Chloro-1-ethyl-[1,2,4]triazolo[4,3...)
Affinity DataIC50: 110nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015779(CHEMBL312449 | 7,8-Dichloro-1-ethyl-[1,2,4]triazol...)
Affinity DataIC50: 110nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015831(CHEMBL310177 | (7,8-Dichloro-1-ethyl-[1,2,4]triazo...)
Affinity DataIC50: 110nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015784(CHEMBL431376 | 1-Ethyl-7-methoxy-[1,2,4]triazolo[4...)
Affinity DataIC50: 140nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015804(CHEMBL73596 | (8-Fluoro-1-methoxy-[1,2,4]triazolo[...)
Affinity DataIC50: 160nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015746(CHEMBL71106 | 1-Ethyl-7-fluoro-[1,2,4]triazolo[4,3...)
Affinity DataIC50: 170nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015797(CHEMBL306850 | Isopropyl-(1-trifluoromethyl-[1,2,4...)
Affinity DataIC50: 170nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015785(CHEMBL73006 | (1-Ethyl-8-fluoro-[1,2,4]triazolo[4,...)
Affinity DataIC50: 180nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015776(CHEMBL72367 | 7-Chloro-[1,2,4]triazolo[4,3-a]quino...)
Affinity DataIC50: 210nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015809(CHEMBL73595 | (6-Chloro-1-ethyl-[1,2,4]triazolo[4,...)
Affinity DataIC50: 220nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015821(CHEMBL421117 | Ethyl-(8-fluoro-1-trifluoromethyl-[...)
Affinity DataIC50: 230nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004571(CHEMBL303198 | CP-66713 | 8-Chloro-1-phenyl-[1,2,4...)
Affinity DataIC50: 270nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015781(CHEMBL72953 | (1-Ethyl-7,8-difluoro-[1,2,4]triazol...)
Affinity DataIC50: 280nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015748(CHEMBL311481 | 8-Fluoro-1-trifluoromethyl-[1,2,4]t...)
Affinity DataIC50: 290nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015756(CHEMBL70701 | 8-Chloro-1-methyl-[1,2,4]triazolo[4,...)
Affinity DataIC50: 350nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015808(CHEMBL70585 | (8-Chloro-[1,2,4]triazolo[4,3-a]quin...)
Affinity DataIC50: 370nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015787(CHEMBL73163 | (8-Chloro-1-ethyl-[1,2,4]triazolo[4,...)
Affinity DataIC50: 380nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
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