Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50001474
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50015743(CHEMBL69034 | Acetic acid 3-[1-(3,6-dihydro-2H-pyr...)
Affinity DataKi:  6nMAssay Description:Ability to displace [3H]- TCP from PCP receptor in tissue homogenate preparation of fresh whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50015738(CHEMBL302321 | 3-[1-(3,6-Dihydro-2H-pyridin-1-yl)-...)
Affinity DataKi:  7nMAssay Description:Ability to displace [3H]TCP from PCP receptor in tissue homogenate preparation of fresh whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50015734(CHEMBL307113 | 1-(1-Thiophen-2-yl-cyclohexyl)-1,2,...)
Affinity DataKi:  12nMAssay Description:Ability to displace [3H]TCP from PCP receptor in tissue homogenate preparation of fresh whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50015741(CHEMBL306450 | 1-[1-(3-Methoxy-phenyl)-cyclohexyl]...)
Affinity DataKi:  33nMAssay Description:Ability to displace [3H]TCP from PCP receptor in tissue homogenate preparation of fresh whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50015732(CHEMBL71302 | 1-(1-Phenyl-cyclohexyl)-1,2,3,6-tetr...)
Affinity DataKi:  37nMAssay Description:Ability to displace [3H]- TCP from PCP receptor in tissue homogenate preparation of fresh whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50015733(CHEMBL71834 | 3-[1-(3,6-Dihydro-2H-pyridin-1-yl)-c...)
Affinity DataKi:  56nMAssay Description:Ability to displace [3H]TCP from PCP receptor in tissue homogenate preparation of fresh whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50015735(CHEMBL307988 | 1-(1-m-Tolyl-cyclohexyl)-1,2,3,6-te...)
Affinity DataKi:  81nMAssay Description:Ability to displace [3H]- TCP from PCP receptor in tissue homogenate preparation of fresh whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50015744(CHEMBL414875 | 1-[1-(3-Methoxymethoxy-phenyl)-cycl...)
Affinity DataKi:  92nMAssay Description:Ability to displace [3H]- TCP from PCP receptor in tissue homogenate preparation of fresh whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50015740(CHEMBL304964 | 1-[1-(3-Vinyl-phenyl)-cyclohexyl]-1...)
Affinity DataKi:  114nMAssay Description:Ability to displace [3H]- TCP from PCP receptor in tissue homogenate preparation of fresh whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50015731(CHEMBL304550 | 1-[1-(3-Methylsulfanyl-phenyl)-cycl...)
Affinity DataKi:  231nMAssay Description:Ability to displace [3H]- TCP from PCP receptor in tissue homogenate preparation of fresh whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50015736(CHEMBL67637 | 1-[1-(3-Fluoro-phenyl)-cyclohexyl]-1...)
Affinity DataKi:  281nMAssay Description:Ability to displace [3H]- TCP from PCP receptor in tissue homogenate preparation of fresh whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50015739(CHEMBL68100 | 3-[1-(3,6-Dihydro-2H-pyridin-1-yl)-c...)
Affinity DataKi:  324nMAssay Description:Ability to displace [3H]- TCP from PCP receptor in tissue homogenate preparation of fresh whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50015730(CHEMBL68156 | 1-[1-(3-Trifluoromethyl-phenyl)-cycl...)
Affinity DataKi:  422nMAssay Description:Ability to displace [3H]- TCP from PCP receptor in tissue homogenate preparation of fresh whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50015742(CHEMBL70943 | 1-[1-(3-[1,3]Dioxolan-2-yl-phenyl)-c...)
Affinity DataKi:  601nMAssay Description:Ability to displace [3H]TCP from PCP receptor in tissue homogenate preparation of fresh whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50015745(CHEMBL71137 | 1-[1-(3-Benzyloxy-phenyl)-cyclohexyl...)
Affinity DataKi:  733nMAssay Description:Ability to displace [3H]TCP from PCP receptor in tissue homogenate preparation of fresh whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50015737(CHEMBL70749 | 1-[1-(3,5-Dimethoxy-phenyl)-cyclohex...)
Affinity DataKi:  8.60E+3nMAssay Description:Ability to displace [3H]TCP from PCP receptor in tissue homogenate preparation of fresh whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed