Compile Data Set for Download or QSAR
Report error Found 69 Enz. Inhib. hit(s) with all data for entry = 50042888
TargetCannabinoid receptor 1(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432712(AM4089 | CHEMBL2348473)
Affinity DataEC50:  450nMAssay Description:Agonist activity at human CB1 receptor transfected in human U2OS cells assessed as beta-arrestin2-GFP aggregation after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432713(CHEMBL2348472)
Affinity DataEC50:  230nMAssay Description:Agonist activity at human CB1 receptor transfected in human U2OS cells assessed as beta-arrestin2-GFP aggregation after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432714(AM4054 | CHEMBL2348462)
Affinity DataEC50:  96nMAssay Description:Agonist activity at human CB1 receptor transfected in human U2OS cells assessed as beta-arrestin2-GFP aggregation after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50169951(AM-411 | (6aR-trans)-3-Adamantan-1-yl-6,6,9-trimet...)
Affinity DataEC50:  1.53E+3nMAssay Description:Agonist activity at human CB1 receptor transfected in human U2OS cells assessed as beta-arrestin2-GFP aggregation after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432712(AM4089 | CHEMBL2348473)
Affinity DataEC50:  8nMAssay Description:Partial agonist activity at human CB1 receptor transfected in HEK293 cells assessed as reduction in forskolin-stimulated cAMP accumulation after 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432714(AM4054 | CHEMBL2348462)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human CB1 receptor transfected in HEK293 cells assessed as reduction in forskolin-stimulated cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataEC50:  1.76E+3nMAssay Description:Agonist activity at human CB1 receptor transfected in human U2OS cells assessed as beta-arrestin2-GFP aggregation after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432712(AM4089 | CHEMBL2348473)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432714(AM4054 | CHEMBL2348462)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432730(CHEMBL2348459)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in HEK293 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50169951(AM-411 | (6aR-trans)-3-Adamantan-1-yl-6,6,9-trimet...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432713(CHEMBL2348472)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432720(CHEMBL2348469)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in HEK293 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432720(CHEMBL2348469)
Affinity DataKi:  8.10nMAssay Description:Displacement of [3H]CP-55940 from mouse CB2 receptor expressed in mouse spleen membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432722(CHEMBL2348467)
Affinity DataKi:  8.60nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432729(CHEMBL2348460)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in HEK293 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432723(CHEMBL2348466)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in HEK293 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432713(CHEMBL2348472)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]CP-55940 from mouse CB2 receptor expressed in mouse spleen membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432714(AM4054 | CHEMBL2348462)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in HEK293 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432714(AM4054 | CHEMBL2348462)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]CP-55940 from mouse CB2 receptor expressed in mouse spleen membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432723(CHEMBL2348466)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432713(CHEMBL2348472)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in HEK293 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432718(CHEMBL2348471)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432720(CHEMBL2348469)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432729(CHEMBL2348460)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]CP-55940 from mouse CB2 receptor expressed in mouse spleen membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432719(CHEMBL2348470)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]CP-55940 from mouse CB2 receptor expressed in mouse spleen membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432728(CHEMBL2348461)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432730(CHEMBL2348459)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]CP-55940 from mouse CB2 receptor expressed in mouse spleen membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432721(CHEMBL2348468)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432724(CHEMBL2348465)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432712(AM4089 | CHEMBL2348473)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]CP-55940 from mouse CB2 receptor expressed in mouse spleen membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432722(CHEMBL2348467)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in HEK293 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432723(CHEMBL2348466)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]CP-55940 from mouse CB2 receptor expressed in mouse spleen membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432722(CHEMBL2348467)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]CP-55940 from mouse CB2 receptor expressed in mouse spleen membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432728(CHEMBL2348461)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]CP-55940 from mouse CB2 receptor expressed in mouse spleen membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432719(CHEMBL2348470)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432728(CHEMBL2348461)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in HEK293 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432717(CHEMBL2348474)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]CP-55940 from mouse CB2 receptor expressed in mouse spleen membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432712(AM4089 | CHEMBL2348473)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in HEK293 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432729(CHEMBL2348460)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432718(CHEMBL2348471)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in HEK293 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432725(CHEMBL2348464)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50169951(AM-411 | (6aR-trans)-3-Adamantan-1-yl-6,6,9-trimet...)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]CP-55940 from mouse CB2 receptor expressed in mouse spleen membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432730(CHEMBL2348459)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432717(CHEMBL2348474)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432717(CHEMBL2348474)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in HEK293 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432721(CHEMBL2348468)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]CP-55940 from mouse CB2 receptor expressed in mouse spleen membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432724(CHEMBL2348465)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in HEK293 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432725(CHEMBL2348464)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]CP-55940 from mouse CB2 receptor expressed in mouse spleen membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50432715(CHEMBL2348476)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
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