Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50042917
TargetCytochrome P450 2C9(Human)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433194(CHEMBL2375587)
Affinity DataIC50: 4.03E+4nMAssay Description:Inhibition of human recombinant CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433194(CHEMBL2375587)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant CYP2D6More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetHistamine H3 receptor(Mouse)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50352090(CHEMBL1824241)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]-iodoproxyfan from histamine H3 receptor in mouse brain cortex after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetHistamine H3 receptor(Mouse)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433200(CHEMBL2375594)
Affinity DataKi:  2.5nMAssay Description:Displacement of [125I]-iodoproxyfan from histamine H3 receptor in mouse brain cortex after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetHistamine H3 receptor(Mouse)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433199(CHEMBL2375595)
Affinity DataKi:  4.30nMAssay Description:Displacement of [125I]-iodoproxyfan from histamine H3 receptor in mouse brain cortex after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetHistamine H3 receptor(Mouse)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433198(CHEMBL2375588)
Affinity DataKi:  6.30nMAssay Description:Displacement of [125I]-iodoproxyfan from histamine H3 receptor in mouse brain cortex after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetHistamine H3 receptor(Mouse)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433194(CHEMBL2375587)
Affinity DataKi:  6.90nMAssay Description:Displacement of [125I]-iodoproxyfan from histamine H3 receptor in mouse brain cortex after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetHistamine H3 receptor(Mouse)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433197(CHEMBL2375597)
Affinity DataKi:  7.60nMAssay Description:Displacement of [125I]-iodoproxyfan from histamine H3 receptor in mouse brain cortex after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetHistamine H3 receptor(Mouse)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433196(CHEMBL2375593)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]-iodoproxyfan from histamine H3 receptor in mouse brain cortex after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetHistamine H3 receptor(Mouse)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433195(CHEMBL2375591)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]-iodoproxyfan from histamine H3 receptor in mouse brain cortex after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed