Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50042901
TargetSerine/threonine-protein kinase pim-3(Human)
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432942(CHEMBL2377721)
Affinity DataIC50: 33nMAssay Description:Inhibition of human full length Pim-3 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432946(CHEMBL2377711)
Affinity DataIC50: 119nMAssay Description:Inhibition of human full length Pim-3 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432946(CHEMBL2377711)
Affinity DataIC50: 230nMAssay Description:Inhibition of human full length Pim-1 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432945(CHEMBL2377716)
Affinity DataIC50: 260nMAssay Description:Inhibition of human full length Pim-3 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432942(CHEMBL2377721)
Affinity DataIC50: 460nMAssay Description:Inhibition of human full length Pim-1 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432947(CHEMBL2377724)
Affinity DataIC50: 470nMAssay Description:Inhibition of human full length Pim-3 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432943(CHEMBL2377718)
Affinity DataIC50: 530nMAssay Description:Inhibition of human full length Pim-3 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432944(CHEMBL2377717)
Affinity DataIC50: 546nMAssay Description:Inhibition of human full length Pim-3 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432943(CHEMBL2377718)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human full length Pim-1 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed