Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 50042569
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50031720((Dofetilide) N-[4-(2-{[2-(4-Methanesulfonylamino-p...)
Affinity DataIC50: 4.10nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427986(CHEMBL2324254)
Affinity DataIC50: 5.10nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427984(CHEMBL2324257)
Affinity DataIC50: 9.90nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427981(CHEMBL2324260)
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427982(CHEMBL2324259)
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427983(CHEMBL2324258)
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427960(CHEMBL2324244)
Affinity DataIC50: 14nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427971(CHEMBL2325208)
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427952(CHEMBL2325199)
Affinity DataIC50: 24nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427974(CHEMBL2325204)
Affinity DataIC50: 24nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427951(CHEMBL2325200)
Affinity DataIC50: 40nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427979(CHEMBL2324262)
Affinity DataIC50: 53nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427959(CHEMBL2324245)
Affinity DataIC50: 60nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427957(2,6-Bis(Phenoxymethyl)Pyridine | CHEMBL2324247)
Affinity DataIC50: 74nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427958(CHEMBL2324246)
Affinity DataIC50: 74nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427950(CHEMBL2325205)
Affinity DataIC50: 86nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427978(CHEMBL2324263)
Affinity DataIC50: 107nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427977(CHEMBL2324264)
Affinity DataIC50: 135nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427953(CHEMBL2324256)
Affinity DataIC50: 146nMAssay Description:Inhibition of human ERG K+ channel expressed in HEK293 cells after 15 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427987(CHEMBL2324243)
Affinity DataIC50: 158nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427953(CHEMBL2324256)
Affinity DataIC50: 170nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427952(CHEMBL2325199)
Affinity DataIC50: 194nMAssay Description:Inhibition of human ERG K+ channel expressed in HEK293 cells after 15 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427988(CHEMBL2324242)
Affinity DataIC50: 208nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427951(CHEMBL2325200)
Affinity DataIC50: 214nMAssay Description:Inhibition of human ERG K+ channel expressed in HEK293 cells after 15 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427976(CHEMBL2325201)
Affinity DataIC50: 285nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427967(CHEMBL2325212)
Affinity DataIC50: 294nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427980(CHEMBL2324261)
Affinity DataIC50: 346nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427973(CHEMBL2325206)
Affinity DataIC50: 371nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427966(CHEMBL2325213)
Affinity DataIC50: 377nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427954(CHEMBL2324251)
Affinity DataIC50: 466nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427969(CHEMBL2325210)
Affinity DataIC50: 554nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427956(CHEMBL2324248)
Affinity DataIC50: 767nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427950(CHEMBL2325205)
Affinity DataIC50: 962nMAssay Description:Inhibition of human ERG K+ channel expressed in HEK293 cells after 15 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427965(CHEMBL2325214)
Affinity DataIC50: 1.16E+3nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427955(2,6-Diphenethylpyridine | CHEMBL2324250)
Affinity DataIC50: 1.61E+3nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427972(CHEMBL2325207)
Affinity DataIC50: 1.99E+3nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427970(CHEMBL2325209)
Affinity DataIC50: 2.91E+3nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427963(CHEMBL2325216)
Affinity DataIC50: 3.90E+3nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427964(CHEMBL2325215)
Affinity DataIC50: 4.02E+3nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427968(CHEMBL2325211)
Affinity DataIC50: 4.34E+3nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427949(CHEMBL2325202)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427985(CHEMBL2324255)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427962(CHEMBL2325217)
Affinity DataIC50: 1.40E+4nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427975(CHEMBL2325203)
Affinity DataIC50: 1.44E+4nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50427961(CHEMBL2324239)
Affinity DataIC50: 3.11E+4nMAssay Description:Displacement of [3H]astemizole from human ERG K+ channel expressed in HEK293 cells by scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed