Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50005275
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM26187(CHEMBL14060 | phenol | US9688816, 2 | α-CA in...)
Affinity DataKd:  1.03E+5nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A/M102H double mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50167939(Benzine | cyclohexatriene | Pyrobenzol | Benzol | ...)
Affinity DataKd:  1.75E+5nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50008558(Toluen | phenylmethane | CHEMBL9113 | Toluol | tol...)
Affinity DataKd:  9.05E+5nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A/M102H double mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50490554(CHEBI:39826 | 2-Allylphenol)
Affinity DataKd:  7.20E+4nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A/M102H double mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM31678(p-nitrophenol)
Affinity DataKd:  3.00E+3nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A/M102H double mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM26187(CHEMBL14060 | phenol | US9688816, 2 | α-CA in...)
Affinity DataKd:  9.10E+4nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A/M102Q double mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50167939(Benzine | cyclohexatriene | Pyrobenzol | Benzol | ...)
Affinity DataKd:  2.70E+4nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A/M102E double mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM31678(p-nitrophenol)
Affinity DataKd:  1.23E+5nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A/M102Q double mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50008567(CHEMBL31561 | para-xylene | 4-xylene | p-dimethylb...)
Affinity DataKd:  4.22E+5nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50167951(ethylbenzene | Aethylbenzol | alpha-methyltoluene ...)
Affinity DataKd:  4.40E+4nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A/M102E double mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50008567(CHEMBL31561 | para-xylene | 4-xylene | p-dimethylb...)
Affinity DataKd:  1.51E+5nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A/M102E double mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50490553(CHEMBL1232569)
Affinity DataKd:  3.17E+5nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A/M102H double mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50167939(Benzine | cyclohexatriene | Pyrobenzol | Benzol | ...)
Affinity DataKd:  4.80E+5nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A/M102H double mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50008558(Toluen | phenylmethane | CHEMBL9113 | Toluol | tol...)
Affinity DataKd:  1.02E+5nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50167951(ethylbenzene | Aethylbenzol | alpha-methyltoluene ...)
Affinity DataKd:  6.80E+4nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50008558(Toluen | phenylmethane | CHEMBL9113 | Toluol | tol...)
Affinity DataKd:  1.56E+5nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A/M102Q double mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM26187(CHEMBL14060 | phenol | US9688816, 2 | α-CA in...)
Affinity DataKd:  1.09E+5nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A/M102E double mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50008558(Toluen | phenylmethane | CHEMBL9113 | Toluol | tol...)
Affinity DataKd:  7.10E+4nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A/M102E double mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed