Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50001430
TargetAdenosine receptor A1(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM82013(NSC_92411 | 8-(2-Amino-4-chlorophenyl)-1,3-dipropy...)
Affinity DataKi:  4.80nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50004575(CHEMBL268071 | Cyclopentyl-(1-trifluoromethyl-[1,2...)
Affinity DataKi:  7.30nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50004566(CHEMBL268431 | 9-chloro-2-(furan-2-yl)-[1,2,4]tria...)
Affinity DataKi:  21nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50015509(CHEMBL301814 | 5-(2-Amino-4-chloro-phenyl)-1,3-dim...)
Affinity DataKi:  310nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM10847(Theophylline (1,3-dimethylxanthine) | 1,3-dimethyl...)
Affinity DataKi:  8.50E+3nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed