Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50042745
TargetC-C chemokine receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50430274(CHEMBL2332935)
Affinity DataIC50: 0.360nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR1 expressed in HEK293 cells after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50430275(CHEMBL2332933)
Affinity DataIC50: 0.360nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR1 expressed in HEK293 cells after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50430280(CHEMBL2332936)
Affinity DataIC50: 0.520nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR1 expressed in HEK293 cells after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50430286(CHEMBL2332931)
Affinity DataIC50: 0.640nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR1 expressed in HEK293 cells after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50430285(CHEMBL2332940)
Affinity DataIC50: 0.790nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR1 expressed in HEK293 cells after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50430284(CHEMBL2332930)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR1 expressed in HEK293 cells after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50430282(CHEMBL2332934)
Affinity DataIC50: 0.960nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR1 expressed in HEK293 cells after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50430283(CHEMBL2332932)
Affinity DataIC50: 0.960nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR1 expressed in HEK293 cells after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50430281(CHEMBL2332941)
Affinity DataIC50: 1.40nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR1 expressed in HEK293 cells after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50430274(CHEMBL2332935)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at CCR1 receptor in human THP1 cells assessed as inhibition of MIP-1alpha-induced chemotaxis after 2 hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50430280(CHEMBL2332936)
Affinity DataIC50: 2.60nMAssay Description:Antagonist activity at CCR1 receptor in human THP1 cells assessed as inhibition of MIP-1alpha-induced chemotaxis after 2 hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50430279(CHEMBL2332937)
Affinity DataIC50: 6nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR1 expressed in HEK293 cells after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50430278(CHEMBL2332938)
Affinity DataIC50: 9nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR1 expressed in HEK293 cells after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50430276(CHEMBL2332942)
Affinity DataIC50: 18nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR1 expressed in HEK293 cells after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50430277(CHEMBL2332939)
Affinity DataIC50: 32nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR1 expressed in HEK293 cells after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50430276(CHEMBL2332942)
Affinity DataIC50: 68nMAssay Description:Antagonist activity at CCR1 receptor in human THP1 cells assessed as inhibition of MIP-1alpha-induced chemotaxis after 2 hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed