Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50042744
TargetSigma non-opioid intracellular receptor 1(Rat)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50430255(CHEMBL240981)
Affinity DataIC50: 1.54E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50430256(NPGI-01 | CHEMBL391409)
Affinity DataIC50: 1.78E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50401370(CHEMBL2205821)
Affinity DataKi:  8.91nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50305342(4-(3'-Fluorophenethyl)-4-azahexacyclo[5.4.1.02,6.0...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50430257(CHEMBL2332492)
Affinity DataKi:  10nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50430259(CHEMBL2332494)
Affinity DataKi:  10nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50288953(CHEMBL1190672 | CHEMBL541347 | 11'N-(3-bromobenzyl...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50401377(CHEMBL2205835)
Affinity DataKi:  20nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50401372(CHEMBL2205819)
Affinity DataKi:  20.9nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50430258(CHEMBL2332493)
Affinity DataKi:  20.9nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50288955(CHEMBL538057 | CHEMBL1189111 | 11'N-benzylspiro[di...)
Affinity DataKi:  67.6nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50288949(CHEMBL552794 | CHEMBL1194508 | 11'N-(4-iodomobenzy...)
Affinity DataKi:  72.4nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50430268(CHEMBL2332502)
Affinity DataKi:  81.3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50430269(CHEMBL2332504)
Affinity DataKi:  85.1nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50430261(CHEMBL2332496)
Affinity DataKi:  97.7nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50401382(CHEMBL2205825)
Affinity DataKi:  102nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50288954(CHEMBL1189234 | CHEMBL538300 | 11-benzyl-11-azahex...)
Affinity DataKi:  102nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50430266(CHEMBL2332501)
Affinity DataKi:  107nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50288950(CHEMBL539310 | CHEMBL1189714 | 11'N-(3-iodobenzyl)...)
Affinity DataKi:  123nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50305343(4-(3'-Fluorophenyl)methyl-4-azahexacyclo[5.4.1.02,...)
Affinity DataKi:  151nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50430267(CHEMBL2332503)
Affinity DataKi:  169nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50430265(CHEMBL2332499)
Affinity DataKi:  181nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50430260(CHEMBL2332495)
Affinity DataKi:  186nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50430264(CHEMBL2332500)
Affinity DataKi:  199nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50288952(11-(3-bromobenzyl)-11-azahexacyclo[5.4.1.02,6.03,1...)
Affinity DataKi:  208nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50430263(CHEMBL2332497)
Affinity DataKi:  269nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Northeast Ohio Medical University

Curated by ChEMBL
LigandPNGBDBM50430262(CHEMBL2332498)
Affinity DataKi:  1.09E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma-1 receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed