Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 8413
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Msa University

LigandPNGBDBM246608(HER2/EGFR dual kinase inhibitor, 5e | 4-{4-[6-(4-(...)
Affinity DataIC50: 1.04E+3nMAssay Description:Protein kinase assays were performed at ambient temperature for 20-40 min (depending on the target) in a final volume of 25 μl according to the fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2017
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Msa University

LigandPNGBDBM246608(HER2/EGFR dual kinase inhibitor, 5e | 4-{4-[6-(4-(...)
Affinity DataIC50: 1.94E+3nMAssay Description:Protein kinase assays were performed at ambient temperature for 20-40 min (depending on the target) in a final volume of 25 μl according to the fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2017
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Msa University

LigandPNGBDBM246607(HER2/EGFR dual kinase inhibitor, 5d)
Affinity DataIC50: 2.09E+3nMAssay Description:Protein kinase assays were performed at ambient temperature for 20-40 min (depending on the target) in a final volume of 25 μl according to the fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2017
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Msa University

LigandPNGBDBM246609(HER2/EGFR dual kinase inhibitor, 7e | (E)-3-(4-Chl...)
Affinity DataIC50: 2.58E+3nMAssay Description:Protein kinase assays were performed at ambient temperature for 20-40 min (depending on the target) in a final volume of 25 μl according to the fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2017
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Msa University

LigandPNGBDBM246607(HER2/EGFR dual kinase inhibitor, 5d)
Affinity DataIC50: 3.98E+3nMAssay Description:Protein kinase assays were performed at ambient temperature for 20-40 min (depending on the target) in a final volume of 25 μl according to the fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2017
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Msa University

LigandPNGBDBM246609(HER2/EGFR dual kinase inhibitor, 7e | (E)-3-(4-Chl...)
Affinity DataIC50: 9.88E+4nMAssay Description:Protein kinase assays were performed at ambient temperature for 20-40 min (depending on the target) in a final volume of 25 μl according to the fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2017
Entry Details Article
PubMed