Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50042440
TargetGlycogen synthase kinase-3 beta(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50426172(Ircinin 1 | CHEMBL483841)
Affinity DataIC50: 794nMAssay Description:Inhibition of human recombinant GSK-3beta using GS2 peptide as substrate and [gamma33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50426172(Ircinin 1 | CHEMBL483841)
Affinity DataIC50: 794nMAssay Description:Inhibition of human recombinant GSK-3beta using GS2 peptide as substrate and [gamma33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50401965(PALINURIN)
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of human recombinant GSK-3alpha using GS2 peptide as substrate and [gamma33P]-ATP after 12 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50401965(PALINURIN)
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of human recombinant GSK-3alpha using GS2 peptide as substrate and [gamma33P]-ATP after 12 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50401965(PALINURIN)
Affinity DataIC50: 1.91E+3nMAssay Description:Inhibition of human recombinant GSK-3beta using GS2 peptide as substrate and [gamma33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50401965(PALINURIN)
Affinity DataIC50: 1.91E+3nMAssay Description:Inhibition of human recombinant GSK-3beta using GS2 peptide as substrate and [gamma33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50426171(Ircinin 2 | CHEMBL483842)
Affinity DataIC50: 2.34E+3nMAssay Description:Inhibition of human recombinant GSK-3beta using GS2 peptide as substrate and [gamma33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50426171(Ircinin 2 | CHEMBL483842)
Affinity DataIC50: 2.34E+3nMAssay Description:Inhibition of human recombinant GSK-3beta using GS2 peptide as substrate and [gamma33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50426173(CHEMBL219346)
Affinity DataIC50: 5.75E+3nMAssay Description:Inhibition of human recombinant GSK-3beta using GS2 peptide as substrate and [gamma33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50426173(CHEMBL219346)
Affinity DataIC50: 5.75E+3nMAssay Description:Inhibition of human recombinant GSK-3beta using GS2 peptide as substrate and [gamma33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50426174(CHEMBL218301)
Affinity DataIC50: 6.17E+3nMAssay Description:Inhibition of human recombinant GSK-3beta using GS2 peptide as substrate and [gamma33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50426174(CHEMBL218301)
Affinity DataIC50: 6.17E+3nMAssay Description:Inhibition of human recombinant GSK-3beta using GS2 peptide as substrate and [gamma33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50401965(PALINURIN)
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of human recombinant CDK5 using histone H1 as substrate and [gamma33P]-ATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50401965(PALINURIN)
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of human recombinant CDK5 using histone H1 as substrate and [gamma33P]-ATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50426175(CHEMBL218931)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant GSK-3beta using GS2 peptide as substrate and [gamma33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50426175(CHEMBL218931)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant GSK-3beta using GS2 peptide as substrate and [gamma33P]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50401965(PALINURIN)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant CDK1 using histone H1 as substrate and [gamma33P]-ATP after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50401965(PALINURIN)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant CDK1 using histone H1 as substrate and [gamma33P]-ATP after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed