Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 50042499
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426906(CHEMBL2323692)
Affinity DataIC50: 8nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426894(CHEMBL2323684)
Affinity DataIC50: 10nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426887(CHEMBL2323695)
Affinity DataIC50: 11nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426906(CHEMBL2323692)
Affinity DataIC50: 12nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426895(CHEMBL2323683)
Affinity DataIC50: 15nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426894(CHEMBL2323684)
Affinity DataIC50: 18nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426895(CHEMBL2323683)
Affinity DataIC50: 20nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426887(CHEMBL2323695)
Affinity DataIC50: 22nMAssay Description:Inhibition of rat SGLT1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426889(CHEMBL2323409)
Affinity DataIC50: 23nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426893(CHEMBL2323405)
Affinity DataIC50: 25nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426893(CHEMBL2323405)
Affinity DataIC50: 42nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426905(CHEMBL2323693)
Affinity DataIC50: 45nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426889(CHEMBL2323409)
Affinity DataIC50: 46nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426888(CHEMBL2323694)
Affinity DataIC50: 50nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426891(CHEMBL2323407)
Affinity DataIC50: 70nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426905(CHEMBL2323693)
Affinity DataIC50: 80nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426892(CHEMBL2323406)
Affinity DataIC50: 98nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426890(CHEMBL2323408)
Affinity DataIC50: 103nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426888(CHEMBL2323694)
Affinity DataIC50: 104nMAssay Description:Inhibition of rat SGLT1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426892(CHEMBL2323406)
Affinity DataIC50: 124nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426891(CHEMBL2323407)
Affinity DataIC50: 151nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426897(CHEMBL2323417)
Affinity DataIC50: 170nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50394533(CHEMBL2159101)
Affinity DataIC50: 183nMAssay Description:Inhibition of rat SGLT1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50394538(CHEMBL2159106)
Affinity DataIC50: 207nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426890(CHEMBL2323408)
Affinity DataIC50: 209nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426899(CHEMBL2323415)
Affinity DataIC50: 217nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50394538(CHEMBL2159106)
Affinity DataIC50: 285nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426897(CHEMBL2323417)
Affinity DataIC50: 319nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426901(CHEMBL2323413)
Affinity DataIC50: 351nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426898(CHEMBL2323416)
Affinity DataIC50: 358nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426887(CHEMBL2323695)
Affinity DataIC50: 371nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426912(CHEMBL2323686)
Affinity DataIC50: 392nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426913(CHEMBL2323685)
Affinity DataIC50: 422nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426907(CHEMBL2323691)
Affinity DataIC50: 446nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426900(CHEMBL2323414)
Affinity DataIC50: 457nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426898(CHEMBL2323416)
Affinity DataIC50: 517nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426899(CHEMBL2323415)
Affinity DataIC50: 608nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426911(CHEMBL2323687)
Affinity DataIC50: 724nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50394550(CHEMBL2160193)
Affinity DataIC50: 738nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426896(CHEMBL2323418)
Affinity DataIC50: 772nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426908(CHEMBL2323690)
Affinity DataIC50: 831nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426909(CHEMBL2323689)
Affinity DataIC50: 931nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426909(CHEMBL2323689)
Affinity DataIC50: 936nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426900(CHEMBL2323414)
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426896(CHEMBL2323418)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426901(CHEMBL2323413)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426887(CHEMBL2323695)
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of rat SGLT2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426904(CHEMBL2323410)
Affinity DataIC50: 1.47E+3nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426910(CHEMBL2323688)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426913(CHEMBL2323685)
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
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