Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 5702
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM50282567(3,4-Dichlorophenyl boronic acid | Phenylboronic ac...)
Affinity DataIC50: 138nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM92722(Phenylboronic acid, 15)
Affinity DataIC50: 238nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM92718(Phenylboronic acid, 10)
Affinity DataIC50: 418nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM92717(Phenylboronic acid, 8)
Affinity DataIC50: 510nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM26139(Phenylboronic acid, 11 | 1-benzothiophen-2-ylboran...)
Affinity DataIC50: 529nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM50282567(3,4-Dichlorophenyl boronic acid | Phenylboronic ac...)
Affinity DataIC50: 1.10E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM92718(Phenylboronic acid, 10)
Affinity DataIC50: 1.40E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM92719(Phenylboronic acid, 12)
Affinity DataIC50: 1.60E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM92721(Phenylboronic acid, 14)
Affinity DataIC50: 1.80E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM92717(Phenylboronic acid, 8)
Affinity DataIC50: 1.97E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM92727(Phenylboronic acid, 20)
Affinity DataIC50: 1.98E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM92726(Phenylboronic acid, 19)
Affinity DataIC50: 2.16E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM26139(Phenylboronic acid, 11 | 1-benzothiophen-2-ylboran...)
Affinity DataIC50: 2.30E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM92719(Phenylboronic acid, 12)
Affinity DataIC50: 2.60E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM92720(Phenylboronic acid, 13)
Affinity DataIC50: 2.70E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM92724(Phenylboronic acid, 17)
Affinity DataIC50: 2.87E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM92723(Phenylboronic acid, 16)
Affinity DataIC50: 2.95E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM92722(Phenylboronic acid, 15)
Affinity DataIC50: 3.20E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM92721(Phenylboronic acid, 14)
Affinity DataIC50: 3.20E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM26132((4-phenylphenyl)boranediol | Phenylboronic acid, 2...)
Affinity DataIC50: 3.55E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM92723(Phenylboronic acid, 16)
Affinity DataIC50: 3.70E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM92724(Phenylboronic acid, 17)
Affinity DataIC50: 3.90E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM92720(Phenylboronic acid, 13)
Affinity DataIC50: 4.10E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM92725(Phenylboronic acid, 18)
Affinity DataIC50: 4.18E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM92725(Phenylboronic acid, 18)
Affinity DataIC50: 4.60E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM92726(Phenylboronic acid, 19)
Affinity DataIC50: 6.30E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM92727(Phenylboronic acid, 20)
Affinity DataIC50: 1.02E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM26140(Phenylboronic acid, 21 | CHEMBL143399 | 1-benzofur...)
Affinity DataIC50: 1.13E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM26140(Phenylboronic acid, 21 | CHEMBL143399 | 1-benzofur...)
Affinity DataIC50: 1.35E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM26996(Phenylboronic acid, 22 | benzeneboronic acid | CHE...)
Affinity DataIC50: 1.48E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM26132((4-phenylphenyl)boranediol | Phenylboronic acid, 2...)
Affinity DataIC50: 1.69E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM26996(Phenylboronic acid, 22 | benzeneboronic acid | CHE...)
Affinity DataIC50: 2.51E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM92728(Phenylboronic acid, 7)
Affinity DataIC50: 3.36E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM92728(Phenylboronic acid, 7)
Affinity DataIC50: 4.15E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Human)
Technical University of Dortmund

LigandPNGBDBM26137((2-phenylphenyl)boranediol | Phenylboronic acid, 2...)
Affinity DataIC50: 5.00E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 2(Human)
Technical University of Dortmund

LigandPNGBDBM26137((2-phenylphenyl)boranediol | Phenylboronic acid, 2...)
Affinity DataIC50: 5.00E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2013
Entry Details Article
PubMed