Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50042355
TargetAdenosine receptor A3(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50424511(CHEMBL2311741)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335734(N-2,6-dibenzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)ac...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335711(N-2,6-bis4-methoxyphenyl)pyrimidin-4-yl)acetamide ...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50424514(CHEMBL2312110)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335731(N-2,6-bis2,4-dimethoxyphenyl)pyrimidin-4-yl)acetam...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50424515(CHEMBL2311746)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50157676(N-(2,6-diphenylpyrimidin-4-yl)acetamide | CHEMBL42...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335734(N-2,6-dibenzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)ac...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50424511(CHEMBL2311741)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335728(N-2,6-bis2-fluorophenyl)pyrimidin-4-yl)acetamide |...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50424512(CHEMBL2312112)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50157676(N-(2,6-diphenylpyrimidin-4-yl)acetamide | CHEMBL42...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50424517(CHEMBL2311743)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50424510(CHEMBL2311745)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50424511(CHEMBL2311741)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]4-(2-[7-Amino-2-(2-furyl) [1,2,4]triazolo[2,3-alpha] [1,3,5]triazin-5-ylamino]ethyl)phenol from human adenosine A2A receptor expr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50424513(CHEMBL2312111)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50424511(CHEMBL2311741)
Affinity DataKi:  68nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50157676(N-(2,6-diphenylpyrimidin-4-yl)acetamide | CHEMBL42...)
Affinity DataKi:  255nMAssay Description:Displacement of [3H]4-(2-[7-Amino-2-(2-furyl) [1,2,4]triazolo[2,3-alpha] [1,3,5]triazin-5-ylamino]ethyl)phenol from human adenosine A2A receptor expr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50424510(CHEMBL2311745)
Affinity DataKi:  375nMAssay Description:Displacement of [3H]4-(2-[7-Amino-2-(2-furyl) [1,2,4]triazolo[2,3-alpha] [1,3,5]triazin-5-ylamino]ethyl)phenol from human adenosine A2A receptor expr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50424518(CHEMBL2311742)
Affinity DataKi:  389nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50424510(CHEMBL2311745)
Affinity DataKi:  494nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50424516(CHEMBL2311744)
Affinity DataKi:  513nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335734(N-2,6-dibenzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)ac...)
Affinity DataKi:  3.35E+3nMAssay Description:Displacement of [3H]4-(2-[7-Amino-2-(2-furyl) [1,2,4]triazolo[2,3-alpha] [1,3,5]triazin-5-ylamino]ethyl)phenol from human adenosine A2A receptor expr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed