Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50040445
TargetPeroxisome proliferator-activated receptor gamma(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394343(CHEMBL516827)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394346(CHEMBL2159605)
Affinity DataEC50:  4.71E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394345(CHEMBL2159606)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394344(CHEMBL2159607)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394343(CHEMBL516827)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394342(CHEMBL458899)
Affinity DataEC50:  4.29E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394341(CHEMBL465800)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50371235(CIPROFIBRATE)
Affinity DataEC50:  900nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394346(CHEMBL2159605)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394345(CHEMBL2159606)
Affinity DataEC50:  3.31E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394344(CHEMBL2159607)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50085041({4-[3-(4-acetyl-3-hydroxy-2-propylphenoxy)propoxy]...)
Affinity DataEC50:  650nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor gamma(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394342(CHEMBL458899)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394341(CHEMBL465800)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50085045(5-((4-((6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydro-...)
Affinity DataEC50:  720nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394346(CHEMBL2159605)
Affinity DataEC50:  1.10E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394345(CHEMBL2159606)
Affinity DataEC50:  1.31E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394344(CHEMBL2159607)
Affinity DataEC50:  3.01E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394343(CHEMBL516827)
Affinity DataEC50:  2.93E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394342(CHEMBL458899)
Affinity DataEC50:  1.56E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394341(CHEMBL465800)
Affinity DataEC50:  2.31E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed