Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50040627
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397290(VUF-10147 | CHEMBL475331)
Affinity DataKi:  0.0513nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50053631(2-(4-methylpiperazin-1-yl)quinoline | 2-(4-Methyl-...)
Affinity DataKi:  0.457nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397307(VUF-10349 | CHEMBL489062)
Affinity DataKi:  1.12nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397291(VUF-10249 | CHEMBL443764)
Affinity DataKi:  1.35nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397284(CHEMBL2169970)
Affinity DataKi:  1.45nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397288(CHEMBL2169966)
Affinity DataKi:  1.62nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397294(VUF-10509 | CHEMBL489271)
Affinity DataKi:  2.69nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397292(VUF-10499 | CHEMBL454890)
Affinity DataKi:  2.82nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397289(CHEMBL2169965)
Affinity DataKi:  2.95nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50060682(2-(4-Methyl-piperazin-1-yl)-quinoxaline | CHEMBL12...)
Affinity DataKi:  4.68nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397283(CHEMBL2169971)
Affinity DataKi:  5.89nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397299(VUF-10350 | CHEMBL489060)
Affinity DataKi:  6.61nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397302(CHEMBL2169890)
Affinity DataKi:  7.41nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397300(VUF-10351 | CHEMBL473302)
Affinity DataKi:  12.0nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397285(CHEMBL2169969)
Affinity DataKi:  13.5nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397296(VUF-10329 | CHEMBL490071)
Affinity DataKi:  13.8nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397293(VUF-10455 | CHEMBL489664)
Affinity DataKi:  14.8nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397308(CHEMBL511699)
Affinity DataKi:  18.2nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM81956(NSC_63211 | CAS_63211 | AMI-098)
Affinity DataKi:  46.8nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397295(VUF-10453 | CHEMBL490072)
Affinity DataKi:  79.4nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397298(VUF-10452 | CHEMBL490073)
Affinity DataKi:  166nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397281(CHEMBL2169973)
Affinity DataKi:  204nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397282(CHEMBL2169972)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397280(CHEMBL2169974)
Affinity DataKi:  331nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397287(CHEMBL2169967)
Affinity DataKi:  407nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397306(CHEMBL2169975)
Affinity DataKi:  468nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397286(CHEMBL2169968)
Affinity DataKi:  537nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397301(VUF-10331 | CHEMBL471712)
Affinity DataKi:  575nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397305(CHEMBL461360)
Affinity DataKi:  2.34E+3nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397304(CHEMBL461729)
Affinity DataKi:  3.55E+3nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397303(CHEMBL462417)
Affinity DataKi:  1.17E+4nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50397297(VUF-10508 | CHEMBL489061)
Affinity DataKi:  1.66E+4nMAssay Description:Displacement of [3H]granisetron from 5HT3A receptor expressed in HEK293 cells after 24 hrs by scintillation counting in presence of quipazineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed