Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50035822
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50014174(CHEMBL289060 | 2-(1H-Imidazol-4-ylmethyl)-4-phenyl...)
Affinity DataKi:  0.990nMAssay Description:In vitro displacement of [3H]ICS-205-930 from 5-hydroxytryptamine 3 receptor in cultured NG-108-15 rat glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50014154(CHEMBL38465 | 2-(5-Methyl-1H-imidazol-4-ylmethyl)-...)
Affinity DataKi:  1.5nMAssay Description:In vitro displacement of [3H]ICS-205-930 from 5-hydroxytryptamine 3 receptor in cultured NG-108-15 rat glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50108392((3-ENDO)-8-METHYL-8-AZABICYCLO[3.2.1]OCT-3-YL 1H-I...)
Affinity DataKi:  2.70nMAssay Description:In vitro displacement of [3H]ICS-205-930 from 5-hydroxytryptamine 3 receptor in cultured NG-108-15 rat glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50013039(CHEMBL40260 | N-[4-(1H-Indol-3-yl)-thiazol-2-ylmet...)
Affinity DataKi:  3.30nMAssay Description:In vitro displacement of [3H]ICS-205-930 from 5-hydroxytryptamine 3 receptor in cultured NG-108-15 rat glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50013043(CHEMBL290938 | 3-[2-(5-Methyl-1H-imidazol-4-ylmeth...)
Affinity DataKi:  10nMAssay Description:In vitro displacement of [3H]ICS-205-930 from 5-hydroxytryptamine 3 receptor in cultured NG-108-15 rat glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50014600(CHEMBL41077 | 3-[2-(1H-Imidazol-4-ylmethyl)-thiazo...)
Affinity DataKi:  14nMAssay Description:In vitro displacement of [3H]ICS-205-930 from 5-hydroxytryptamine 3 receptor in cultured NG-108-15 rat glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM85330(NSC_68647 | CAS_68647 | ONDANSETRON | Ondansetron ...)
Affinity DataKi:  16nMAssay Description:In vitro displacement of [3H]ICS-205-930 from 5-hydroxytryptamine 3 receptor in cultured NG-108-15 rat glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50014601(CHEMBL288435 | 2-(2-Methyl-1H-imidazol-4-ylmethyl)...)
Affinity DataKi:  226nMAssay Description:In vitro displacement of [3H]ICS-205-930 from 5-hydroxytryptamine 3 receptor in cultured NG-108-15 rat glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50013045(CHEMBL290266 | 3-[2-(2-Methyl-imidazol-1-ylmethyl)...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro displacement of [3H]ICS-205-930 from 5-hydroxytryptamine 3 receptor in cultured NG-108-15 rat glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50014406(CHEMBL266591 | 2-Methyl-5-hydroxytryptamine | 2-Me...)
Affinity DataKi:  1.22E+3nMAssay Description:In vitro displacement of [3H]ICS-205-930 from 5-hydroxytryptamine 3 receptor in cultured NG-108-15 rat glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed