Compile Data Set for Download or QSAR
Report error Found 89 Enz. Inhib. hit(s) with all data for entry = 50042141
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421255(CHEMBL2087873)
Affinity DataIC50: 5nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421256(CHEMBL2087874)
Affinity DataIC50: 10nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421257(CHEMBL2087875)
Affinity DataIC50: 10nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421279(CHEMBL2087655)
Affinity DataIC50: 20nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421284(CHEMBL2087660)
Affinity DataIC50: 20nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421289(CHEMBL2087666)
Affinity DataIC50: 20nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421286(CHEMBL2087662)
Affinity DataIC50: 20nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50204587((S)-6-(4-(2-(dimethylamino)ethoxy)phenyl)-5-phenyl...)
Affinity DataIC50: 30nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421254(CHEMBL2087872)
Affinity DataIC50: 40nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421278(CHEMBL2087654)
Affinity DataIC50: 40nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421287(CHEMBL2087664)
Affinity DataIC50: 40nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421282(CHEMBL2087658)
Affinity DataIC50: 60nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421281(CHEMBL2087657)
Affinity DataIC50: 80nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421276(CHEMBL2087652)
Affinity DataIC50: 90nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421275(CHEMBL2087651)
Affinity DataIC50: 100nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421280(CHEMBL2087656)
Affinity DataIC50: 160nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421253(CHEMBL2087871)
Affinity DataIC50: 160nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421270(CHEMBL2087671)
Affinity DataIC50: 160nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421285(CHEMBL2087661)
Affinity DataIC50: 180nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421288(CHEMBL2087665)
Affinity DataIC50: 190nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421283(CHEMBL2087659)
Affinity DataIC50: 230nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421291(CHEMBL2087668)
Affinity DataIC50: 240nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421274(CHEMBL2087650)
Affinity DataIC50: 250nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421277(CHEMBL2087653)
Affinity DataIC50: 300nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421273(CHEMBL2087649)
Affinity DataIC50: 350nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421269(CHEMBL2087670)
Affinity DataIC50: 390nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421262(CHEMBL2087880)
Affinity DataIC50: 410nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421293(CHEMBL2087881)
Affinity DataIC50: 420nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421263(CHEMBL2087882)
Affinity DataIC50: 460nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421290(CHEMBL2087667)
Affinity DataIC50: 500nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421272(CHEMBL2087648)
Affinity DataIC50: 550nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421261(CHEMBL2087879)
Affinity DataIC50: 550nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421271(CHEMBL2087647)
Affinity DataIC50: 620nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421264(CHEMBL2087883)
Affinity DataIC50: 780nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421265(CHEMBL2087884)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421259(CHEMBL2087877)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421294(CHEMBL2087663)
Affinity DataIC50: 2.05E+3nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421258(CHEMBL2087876)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM17715(N-[(2S)-oxolan-2-ylmethyl]-2,3-diphenylfuro[2,3-b]...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421260(CHEMBL2087878)
Affinity DataIC50: 7.16E+3nMAssay Description:Inhibition of ACK1 in mouse C8 cells assessed as decrease in cell viability after 20 to 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421256(CHEMBL2087874)
Affinity DataKi:  0.200nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 expressed in baculovirus infected Hi5 cells assessed as inhibition of autophosphorylation after 2 hrs by EL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421257(CHEMBL2087875)
Affinity DataKi:  0.300nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 expressed in baculovirus infected Hi5 cells assessed as inhibition of autophosphorylation after 2 hrs by EL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421255(CHEMBL2087873)
Affinity DataKi:  0.300nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 expressed in baculovirus infected Hi5 cells assessed as inhibition of autophosphorylation after 2 hrs by EL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421278(CHEMBL2087654)
Affinity DataKi:  2nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 expressed in baculovirus infected Hi5 cells assessed as inhibition of autophosphorylation after 2 hrs by EL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421286(CHEMBL2087662)
Affinity DataKi:  2nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 expressed in baculovirus infected Hi5 cells assessed as inhibition of autophosphorylation after 2 hrs by EL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421276(CHEMBL2087652)
Affinity DataKi:  2nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 expressed in baculovirus infected Hi5 cells assessed as inhibition of autophosphorylation after 2 hrs by EL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421287(CHEMBL2087664)
Affinity DataKi:  3nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 expressed in baculovirus infected Hi5 cells assessed as inhibition of autophosphorylation after 2 hrs by EL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421261(CHEMBL2087879)
Affinity DataKi:  4nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 expressed in baculovirus infected Hi5 cells assessed as inhibition of autophosphorylation after 2 hrs by EL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421254(CHEMBL2087872)
Affinity DataKi:  4nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 expressed in baculovirus infected Hi5 cells assessed as inhibition of autophosphorylation after 2 hrs by EL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50421277(CHEMBL2087653)
Affinity DataKi:  4nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 expressed in baculovirus infected Hi5 cells assessed as inhibition of autophosphorylation after 2 hrs by EL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
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