Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50040669
TargetAngiotensin-converting enzyme(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398088(CHEMBL2097001)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of ACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398076(CHEMBL2182011)
Affinity DataIC50: 300nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398075(CHEMBL2182012)
Affinity DataIC50: 300nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398079(CHEMBL2182018)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398078(CHEMBL2182019)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398081(CHEMBL2182013)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398075(CHEMBL2182012)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398080(CHEMBL2182014)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398085(CHEMBL2182017)
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398086(CHEMBL2182016)
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398084(CHEMBL2182020)
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProthrombin(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398077(CHEMBL1256178)
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of thrombin assessed as hydrolysis of H-D-Pro-L-Phe-L-Arg-p-nitroanilide incubated for 2 hrs measured for 20 mins by microplate reader ana...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProthrombin(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398079(CHEMBL2182018)
Affinity DataIC50: 9.20E+4nMAssay Description:Inhibition of thrombin assessed as hydrolysis of H-D-Pro-L-Phe-L-Arg-p-nitroanilide incubated for 2 hrs measured for 20 mins by microplate reader ana...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPlasminogen(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398078(CHEMBL2182019)
Affinity DataIC50: 9.90E+4nMAssay Description:Inhibition of plasmin assessed as hydrolysis of H-D-Val-L-Leu-L-Lys-p-nitroanilide incubated for 2 hrs measured for 20 mins by microplate reader anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProthrombin(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398078(CHEMBL2182019)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of thrombin assessed as hydrolysis of H-D-Pro-L-Phe-L-Arg-p-nitroanilide incubated for 2 hrs measured for 20 mins by microplate reader ana...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCathepsin G(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398079(CHEMBL2182018)
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of cathepsin G assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Phe-p-nitroanilide incubated for 2 hrs measured for 20 mins by microplate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398082(CHEMBL2182022)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398083(CHEMBL2182021)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398087(CHEMBL2182015)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPlasminogen(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398077(CHEMBL1256178)
Affinity DataIC50: 2.40E+5nMAssay Description:Inhibition of plasmin assessed as hydrolysis of H-D-Val-L-Leu-L-Lys-p-nitroanilide incubated for 2 hrs measured for 20 mins by microplate reader anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCathepsin G(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398077(CHEMBL1256178)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of cathepsin G assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Phe-p-nitroanilide incubated for 2 hrs measured for 20 mins by microplate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398075(CHEMBL2182012)
Affinity DataKi:  3.50E+3nMAssay Description:Uncompetitive inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398081(CHEMBL2182013)
Affinity DataKi:  4.00E+3nMAssay Description:Uncompetitive inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398080(CHEMBL2182014)
Affinity DataKi:  5.00E+3nMAssay Description:Uncompetitive inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398079(CHEMBL2182018)
Affinity DataKi:  1.30E+4nMAssay Description:Noncompetitive inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398078(CHEMBL2182019)
Affinity DataKi:  1.80E+4nMAssay Description:Noncompetitive inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed