Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50040667
TargetP2Y purinoceptor 1(Rat)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50398072(CHEMBL2181943)
Affinity DataEC50:  28nMAssay Description:Agonist activity at rat P2Y1R assessed as glucose-dependent insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50118242([({[(2R,3S,4R,5R)-5-[6-amino-2-(methylsulfanyl)-9H...)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at turkey P2Y1R expressed in 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50398066(CHEMBL2181941)
Affinity DataEC50:  34nMAssay Description:Agonist activity at turkey P2Y1R expressed in 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50398067(CHEMBL2181940)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at turkey P2Y1R expressed in 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50398068(CHEMBL2181936)
Affinity DataEC50:  140nMAssay Description:Agonist activity at turkey P2Y1R expressed in 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50398069(CHEMBL2181935)
Affinity DataEC50:  190nMAssay Description:Agonist activity at turkey P2Y1R expressed in 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50398070(CHEMBL2181938)
Affinity DataEC50:  960nMAssay Description:Agonist activity at turkey P2Y1R expressed in 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50398071(CHEMBL2181939)
Affinity DataEC50:  220nMAssay Description:Agonist activity at turkey P2Y1R expressed in 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Rat)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50366480(ATP | ADENOSINE TRIPHOSPHATE)
Affinity DataEC50:  200nMAssay Description:Agonist activity at rat P2Y1R expressed in HEK293 cells assessed as release of intracellular calcium by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Rat)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50398072(CHEMBL2181943)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at rat P2Y1R expressed in HEK293 cells assessed as release of intracellular calcium by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed