Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50040157
TargetP2Y purinoceptor 1(Human)
National Institutes of Health

Curated by ChEMBL
LigandPNGBDBM50390018(CHEMBL2071539)
Affinity DataIC50: 130nMAssay Description:Antagonist activity at human P2Y1R expressed in human 1321N1 cells assessed as inhibition of 2-MeSADP-induced increase in intracellular inositol phos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
National Institutes of Health

Curated by ChEMBL
LigandPNGBDBM59704(cid_1188014 | SMR000078689 | 4-({[(3,4-dichlorophe...)
Affinity DataIC50: 140nMAssay Description:Antagonist activity at human P2Y1R expressed in human 1321N1 cells assessed as inhibition of 2-MeSADP-induced increase in intracellular inositol phos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
National Institutes of Health

Curated by ChEMBL
LigandPNGBDBM50390013(CHEMBL2071529)
Affinity DataKi:  6.00E+3nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
National Institutes of Health

Curated by ChEMBL
LigandPNGBDBM50390014(CHEMBL2071530)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
National Institutes of Health

Curated by ChEMBL
LigandPNGBDBM59704(cid_1188014 | SMR000078689 | 4-({[(3,4-dichlorophe...)
Affinity DataKi:  1.30E+4nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
National Institutes of Health

Curated by ChEMBL
LigandPNGBDBM50390015(CHEMBL2071532)
Affinity DataKi:  2.70E+4nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
National Institutes of Health

Curated by ChEMBL
LigandPNGBDBM50390016(CHEMBL2071534)
Affinity DataKi:  4.20E+4nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
National Institutes of Health

Curated by ChEMBL
LigandPNGBDBM50390017(CHEMBL2071537)
Affinity DataKi:  4.50E+4nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed