Compile Data Set for Download or QSAR
Report error Found 79 Enz. Inhib. hit(s) with all data for entry = 5716
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92800BDBM92800(Bisanilinopyrimidine, 3o | US9249124, 16)
Affinity DataIC50: 0.800nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92810BDBM92810(Bisanilinopyrimidine, 6c | US9249124, 26)
Affinity DataIC50: 2nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 87054BDBM87054(Bisanilinopyrimidine, 6i | Bisanilinopyrimidine in...)
Affinity DataIC50: 2.10nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 87053BDBM87053(Bisanilinopyrimidine, 3l | Bisanilinopyrimidine in...)
Affinity DataIC50: 2.5nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92844BDBM92844(Bisanilinopyrimidine, 12b | US9249124, 60)
Affinity DataIC50: 2.90nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92846BDBM92846(Bisanilinopyrimidine, 12d | US9249124, 62)
Affinity DataIC50: 3nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92843BDBM92843(Bisanilinopyrimidine, 12a | US9249124, 59)
Affinity DataIC50: 3.10nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92805BDBM92805(Bisanilinopyrimidine, 4d | US9249124, 21)
Affinity DataIC50: 3.17nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92817BDBM92817(Bisanilinopyrimidine, 6j | US9249124, 33)
Affinity DataIC50: 3.30nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 87052BDBM87052(Bisanilinopyrimidine, 6a | Bisanilinopyrimidine in...)
Affinity DataIC50: 3.70nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92799BDBM92799(Bisanilinopyrimidine, 3n | US9249124, 15)
Affinity DataIC50: 3.90nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92812BDBM92812(Bisanilinopyrimidine, 6e | US9249124, 28)
Affinity DataIC50: 4nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92827BDBM92827(Bisanilinopyrimidine, 6t)
Affinity DataIC50: 4.5nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92803BDBM92803(Bisanilinopyrimidine, 3r | US9249124, 19)
Affinity DataIC50: 5.10nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 87048BDBM87048(Bisanilinopyrimidine, 1 | Bisanilinopyrimidine inh...)
Affinity DataIC50: 6.10nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92818BDBM92818(Bisanilinopyrimidine, 6k)
Affinity DataIC50: 6.60nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92825BDBM92825(Bisanilinopyrimidine, 6r | US9249124, 41)
Affinity DataIC50: 8.5nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 87047BDBM87047(Bisanilinopyrimidine, 3h | Bisanilinopyrimidine in...)
Affinity DataIC50: 10nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAurora kinase B(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92841BDBM92841(Bisanilinopyrimidine, 9m | US9249124, 57)
Affinity DataIC50: 10.7nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 16011BDBM16011(Bisanilinopyrimidine, 3m | 2-{[5-fluoro-2-(phenyla...)
Affinity DataIC50: 11.3nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92840BDBM92840(Bisanilinopyrimidine, 9l | US9249124, 56)
Affinity DataIC50: 12.3nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92841BDBM92841(Bisanilinopyrimidine, 9m | US9249124, 57)
Affinity DataIC50: 14.4nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92845BDBM92845(Bisanilinopyrimidine, 12c | US9249124, 61)
Affinity DataIC50: 17.3nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92830BDBM92830(Bisanilinopyrimidine, 9c | US9249124, 46)
Affinity DataIC50: 18nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92802BDBM92802(Bisanilinopyrimidine, 3q | US9249124, 18)
Affinity DataIC50: 18.3nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92822BDBM92822(Bisanilinopyrimidine, 6o)
Affinity DataIC50: 18.7nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92801BDBM92801(Bisanilinopyrimidine, 3p | US9249124, 17)
Affinity DataIC50: 19.9nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92842BDBM92842(Bisanilinopyrimidine, 9n | US9249124, 58)
Affinity DataIC50: 21.2nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92838BDBM92838(Bisanilinopyrimidine, 9j | US9249124, 54)
Affinity DataIC50: 21.4nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92839BDBM92839(Bisanilinopyrimidine, 9k | US9249124, 55)
Affinity DataIC50: 23.2nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92838BDBM92838(Bisanilinopyrimidine, 9j | US9249124, 54)
Affinity DataIC50: 25.6nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92835BDBM92835(Bisanilinopyrimidine, 9h | US9249124, 51)
Affinity DataIC50: 27nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 87051BDBM87051(Bisanilinopyrimidine, 6d | Bisanilinopyrimidine in...)
Affinity DataIC50: 28nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92829BDBM92829(Bisanilinopyrimidine, 9b | US9249124, 44)
Affinity DataIC50: 28.1nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92839BDBM92839(Bisanilinopyrimidine, 9k | US9249124, 55)
Affinity DataIC50: 30nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92836BDBM92836(Bisanilinopyrimidine, 6p | US9249124, 52)
Affinity DataIC50: 30.2nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92820BDBM92820(Bisanilinopyrimidine, 6m | US9249124, 36)
Affinity DataIC50: 35nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 87050BDBM87050(Bisanilinopyrimidine, 6h | Bisanilinopyrimidine in...)
Affinity DataIC50: 35.1nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92793BDBM92793(Bisanilinopyrimidine, 3g)
Affinity DataIC50: 38.2nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAurora kinase B(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92840BDBM92840(Bisanilinopyrimidine, 9l | US9249124, 56)
Affinity DataIC50: 40.4nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 87055BDBM87055(Bisanilinopyrimidine, 6n | Bisanilinopyrimidine in...)
Affinity DataIC50: 43nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAurora kinase B(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92837BDBM92837(Bisanilinopyrimidine, 9i | US9249124, 53)
Affinity DataIC50: 43.3nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92831BDBM92831(Bisanilinopyrimidine, 9d | US9249124, 47)
Affinity DataIC50: 44.9nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92813BDBM92813(Bisanilinopyrimidine, 6f | US9249124, 29)
Affinity DataIC50: 46.6nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92826BDBM92826(Bisanilinopyrimidine, 6s | US9249124, 42)
Affinity DataIC50: 50.2nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92836BDBM92836(Bisanilinopyrimidine, 6p | US9249124, 52)
Affinity DataIC50: 50.2nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92842BDBM92842(Bisanilinopyrimidine, 9n | US9249124, 58)
Affinity DataIC50: 56.6nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 16005BDBM16005(2-[(2-{[4-(morpholin-4-yl)phenyl]amino}pyrimidin-4...)
Affinity DataIC50: 57.6nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 92832BDBM92832(Bisanilinopyrimidine, 9e)
Affinity DataIC50: 71.2nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandChemical structure of BindingDB Monomer ID 15991BDBM15991(2-{[2-(phenylamino)pyrimidin-4-yl]amino}benzoic ac...)
Affinity DataIC50: 79.4nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2013
Entry Details Article
PubMed
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