Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50040414
TargetMu-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50001709(CHEMBL558140 | CHEMBL140278 | 4-cyclopropylmethyl-...)
Affinity DataEC50:  1.20nMAssay Description:Inverse agonist activity at human recombinant mu opioid receptor expressed in CHO cells after 3 hrs by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50297506(l7-(cyclopropylmethyl)-3,l4-dihydroxy-6beta-((meth...)
Affinity DataEC50:  2.60nMAssay Description:Inverse agonist activity at human recombinant mu opioid receptor expressed in CHO cells after 3 hrs by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of New England

Curated by ChEMBL
LigandPNGBDBM50297506(l7-(cyclopropylmethyl)-3,l4-dihydroxy-6beta-((meth...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed