Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50040500
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Massachusetts General Hospital

Curated by ChEMBL
LigandPNGBDBM50395121(CHEMBL2163548)
Affinity DataIC50: 3.80E+3nMAssay Description:Displacement of [3H]R-(-)-14 from human FLAG-tagged alpha1 GABA A receptor expressed in HEK293S cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Human)
Massachusetts General Hospital

Curated by ChEMBL
LigandPNGBDBM50395121(CHEMBL2163548)
Affinity DataIC50: 3.90E+3nMAssay Description:Displacement of [3H]R-(-)-14 from human FLAG-tagged beta3 GABA A receptor expressed in HEK293S cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Human)
Massachusetts General Hospital

Curated by ChEMBL
LigandPNGBDBM50055935(5-ethyl-5-(pentan-2-yl)pyrimidine-2,4,6(1H,3H,5H)-...)
Affinity DataIC50: 8.80E+4nMAssay Description:Displacement of [3H]R-(-)-14 from human FLAG-tagged beta3 GABA A receptor expressed in HEK293S cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Massachusetts General Hospital

Curated by ChEMBL
LigandPNGBDBM50395120(CHEMBL2163549)
Affinity DataIC50: 1.20E+5nMAssay Description:Displacement of [3H]R-(-)-14 from human FLAG-tagged alpha1 GABA A receptor expressed in HEK293S cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Human)
Massachusetts General Hospital

Curated by ChEMBL
LigandPNGBDBM50395120(CHEMBL2163549)
Affinity DataIC50: 1.70E+5nMAssay Description:Displacement of [3H]R-(-)-14 from human FLAG-tagged beta3 GABA A receptor expressed in HEK293S cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Massachusetts General Hospital

Curated by ChEMBL
LigandPNGBDBM50055935(5-ethyl-5-(pentan-2-yl)pyrimidine-2,4,6(1H,3H,5H)-...)
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of [3H]R-(-)-14 from human FLAG-tagged alpha1 GABA A receptor expressed in HEK293S cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed