Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50039911
TargetCruzipain(Trypanosoma cruzi)
Instituto De Tecnologia Em F£Rmacos - Farmanguinhos

Curated by ChEMBL
LigandPNGBDBM50386184(CHEMBL2042801)
Affinity DataIC50: 600nMAssay Description:Inhibition of Trypanosoma cruzi cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
Instituto De Tecnologia Em F£Rmacos - Farmanguinhos

Curated by ChEMBL
LigandPNGBDBM50386183(CHEMBL507837)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
Instituto De Tecnologia Em F£Rmacos - Farmanguinhos

Curated by ChEMBL
LigandPNGBDBM50386181(CHEMBL2042793)
Affinity DataIC50: 4.47E+4nMAssay Description:Inhibition of Trypanosoma cruzi C-terminally truncated cruzain expressed in Escherichia coli using Z-Phe-Arg-AMC as substrate incubated for 5 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
Instituto De Tecnologia Em F£Rmacos - Farmanguinhos

Curated by ChEMBL
LigandPNGBDBM50386179(CHEMBL2042791)
Affinity DataIC50: 4.59E+4nMAssay Description:Inhibition of Trypanosoma cruzi C-terminally truncated cruzain expressed in Escherichia coli using Z-Phe-Arg-AMC as substrate incubated for 5 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
Instituto De Tecnologia Em F£Rmacos - Farmanguinhos

Curated by ChEMBL
LigandPNGBDBM50386185(CHEMBL2042780)
Affinity DataIC50: 5.22E+4nMAssay Description:Inhibition of Trypanosoma cruzi C-terminally truncated cruzain expressed in Escherichia coli using Z-Phe-Arg-AMC as substrate incubated for 5 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
Instituto De Tecnologia Em F£Rmacos - Farmanguinhos

Curated by ChEMBL
LigandPNGBDBM50386186(CHEMBL2042788)
Affinity DataIC50: 7.48E+4nMAssay Description:Inhibition of Trypanosoma cruzi C-terminally truncated cruzain expressed in Escherichia coli using Z-Phe-Arg-AMC as substrate incubated for 5 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
Instituto De Tecnologia Em F£Rmacos - Farmanguinhos

Curated by ChEMBL
LigandPNGBDBM50386180(CHEMBL2042792)
Affinity DataIC50: 8.39E+4nMAssay Description:Inhibition of Trypanosoma cruzi C-terminally truncated cruzain expressed in Escherichia coli using Z-Phe-Arg-AMC as substrate incubated for 5 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
Instituto De Tecnologia Em F£Rmacos - Farmanguinhos

Curated by ChEMBL
LigandPNGBDBM50386182(CHEMBL2042797)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi C-terminally truncated cruzain expressed in Escherichia coli using Z-Phe-Arg-AMC as substrate incubated for 5 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed