Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50039962
TargetSodium-dependent dopamine transporter(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50386904(CHEMBL2048526)
Affinity DataKd:  1.20nMAssay Description:Binding affinity to DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataKi:  2.42nMAssay Description:Displacement of [125I]IPT from DAT overexpressed in LLC-PK1 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSodium-dependent dopamine transporter(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50386906(CHEMBL2048520)
Affinity DataKi:  2.64nMAssay Description:Displacement of [125I]IPT from DAT overexpressed in LLC-PK1 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50386905(CHEMBL2048519)
Affinity DataKi:  3.79nMAssay Description:Displacement of [125I]IPT from DAT overexpressed in LLC-PK1 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50386907(CHEMBL2048521)
Affinity DataKi:  4.63nMAssay Description:Displacement of [125I]IPT from DAT overexpressed in LLC-PK1 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50386903(CHEMBL559741)
Affinity DataKi:  12nMAssay Description:Binding affinity to DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50386910(CHEMBL2048524)
Affinity DataKi:  18.3nMAssay Description:Displacement of [125I]IPT from DAT overexpressed in LLC-PK1 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50386911(CHEMBL2048525)
Affinity DataKi:  26.9nMAssay Description:Displacement of [125I]IPT from DAT overexpressed in LLC-PK1 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50386909(CHEMBL2048523)
Affinity DataKi:  135nMAssay Description:Displacement of [125I]IPT from DAT overexpressed in LLC-PK1 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50386908(CHEMBL2048522)
Affinity DataKi:  699nMAssay Description:Displacement of [125I]IPT from DAT overexpressed in LLC-PK1 cell membrane by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed