Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50039797
TargetSolute carrier family 12 member 5(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50384300(CHEMBL2030661)
Affinity DataIC50: 200nMAssay Description:Inhibition of rat KCC2 expressed in human Sk-Hep cells assessed as induction off Rb+ flux by atomic absorption spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSolute carrier family 12 member 5(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50384302(CHEMBL2030663)
Affinity DataIC50: 200nMAssay Description:Inhibition of rat KCC2 expressed in human Sk-Hep cells assessed as induction off Rb+ flux by atomic absorption spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSolute carrier family 12 member 5(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50384298(CHEMBL2030659)
Affinity DataIC50: 300nMAssay Description:Inhibition of rat KCC2 expressed in human Sk-Hep cells assessed as induction off Rb+ flux by atomic absorption spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSolute carrier family 12 member 5(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50384301(CHEMBL2030662)
Affinity DataIC50: 300nMAssay Description:Inhibition of rat KCC2 expressed in human Sk-Hep cells assessed as induction off Rb+ flux by atomic absorption spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSolute carrier family 12 member 5(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50384307(CHEMBL2030669)
Affinity DataIC50: 600nMAssay Description:Inhibition of rat KCC2 expressed in human Sk-Hep cells assessed as induction off Rb+ flux by atomic absorption spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSolute carrier family 12 member 5(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50315350((+/-)-benzyl 1-acetyl-2-benzylpyrrolidine-2-carbox...)
Affinity DataIC50: 800nMAssay Description:Inhibition of rat KCC2 expressed in human Sk-Hep cells assessed as induction off Rb+ flux by atomic absorption spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSolute carrier family 12 member 5(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50384305(CHEMBL2030667)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat KCC2 expressed in human Sk-Hep cells assessed as induction off Rb+ flux by atomic absorption spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSolute carrier family 12 member 5(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50384304(CHEMBL2030665)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rat KCC2 expressed in human Sk-Hep cells assessed as induction off Rb+ flux by atomic absorption spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSolute carrier family 12 member 5(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50384306(CHEMBL2030668)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of rat KCC2 expressed in human Sk-Hep cells assessed as induction off Rb+ flux by atomic absorption spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSolute carrier family 12 member 5(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50384308(CHEMBL2030666)
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of rat KCC2 expressed in human Sk-Hep cells assessed as induction off Rb+ flux by atomic absorption spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSolute carrier family 12 member 5(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50384303(CHEMBL2030664)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of rat KCC2 expressed in human Sk-Hep cells assessed as induction off Rb+ flux by atomic absorption spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSolute carrier family 12 member 5(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50384299(CHEMBL2030660)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of rat KCC2 expressed in human Sk-Hep cells assessed as induction off Rb+ flux by atomic absorption spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed