Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50039761
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383600(CHEMBL2032415)
Affinity DataIC50: 13nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383573(CHEMBL2029489)
Affinity DataIC50: 15nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383581(CHEMBL2029482)
Affinity DataIC50: 15nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383579(CHEMBL2029483)
Affinity DataIC50: 16nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383604(CHEMBL2029481)
Affinity DataIC50: 23nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383598(CHEMBL2032417)
Affinity DataIC50: 24nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383599(CHEMBL2032416)
Affinity DataIC50: 26nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383578(CHEMBL2029484)
Affinity DataIC50: 29nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383591(CHEMBL2032422)
Affinity DataIC50: 36nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383590(CHEMBL2032424)
Affinity DataIC50: 37nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50312718(torcetrapib | CHEMBL479527)
Affinity DataIC50: 39nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383588(CHEMBL2029379)
Affinity DataIC50: 40nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383592(CHEMBL2032421)
Affinity DataIC50: 42nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383576(CHEMBL2029486)
Affinity DataIC50: 44nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383593(CHEMBL2032420)
Affinity DataIC50: 47nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383589(CHEMBL2032425)
Affinity DataIC50: 47nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383597(CHEMBL2032418)
Affinity DataIC50: 48nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383575(CHEMBL2029487)
Affinity DataIC50: 49nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383587(CHEMBL2032426)
Affinity DataIC50: 54nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383596(CHEMBL2032419)
Affinity DataIC50: 55nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383585(CHEMBL2029477)
Affinity DataIC50: 56nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383572(CHEMBL2029490)
Affinity DataIC50: 56nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383602(CHEMBL2032413)
Affinity DataIC50: 57nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383580(CHEMBL2032423)
Affinity DataIC50: 58nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383582(CHEMBL2029480)
Affinity DataIC50: 61nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383595(CHEMBL2032427)
Affinity DataIC50: 74nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383568(CHEMBL2029494)
Affinity DataIC50: 78nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383570(CHEMBL2029492)
Affinity DataIC50: 151nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383571(CHEMBL2029491)
Affinity DataIC50: 162nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383586(CHEMBL2029476)
Affinity DataIC50: 187nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383603(CHEMBL2032412)
Affinity DataIC50: 195nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383569(CHEMBL2029493)
Affinity DataIC50: 218nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383567(CHEMBL2029496)
Affinity DataIC50: 327nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383601(CHEMBL2032414)
Affinity DataIC50: 2.31E+3nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383574(CHEMBL2029488)
Affinity DataIC50: 2.35E+3nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383577(CHEMBL2029485)
Affinity DataIC50: 3.79E+3nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383594(CHEMBL2029495)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383583(CHEMBL2029479)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50383584(CHEMBL2029478)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CETP in human plasma assessed as transfer of fluorescently labelled cholesteryl ester to VLDL by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed