Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50004642
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50485177(CHEMBL2036478)
Affinity DataIC50: 4nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts using Ac-Arg-Gly-Lys(Ac)-AMC substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50485179(CHEMBL2036476)
Affinity DataIC50: 5nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts using Ac-Arg-Gly-Lys(Ac)-AMC substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50485172(CHEMBL2036482)
Affinity DataIC50: 7nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts using Ac-Arg-Gly-Lys(Ac)-AMC substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50485174(CHEMBL2036479)
Affinity DataIC50: 19nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts using Ac-Arg-Gly-Lys(Ac)-AMC substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50485176(CHEMBL2036475)
Affinity DataIC50: 23nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts using Ac-Arg-Gly-Lys(Ac)-AMC substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50485178(CHEMBL2036469)
Affinity DataIC50: 31nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts using Ac-Arg-Gly-Lys(Ac)-AMC substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50485173(CHEMBL2036470)
Affinity DataIC50: 41nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts using Ac-Arg-Gly-Lys(Ac)-AMC substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50485167(CHEMBL2036473)
Affinity DataIC50: 49nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts using Ac-Arg-Gly-Lys(Ac)-AMC substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 67nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts using Ac-Arg-Gly-Lys(Ac)-AMC substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50485168(CHEMBL2036474)
Affinity DataIC50: 86nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts using Ac-Arg-Gly-Lys(Ac)-AMC substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50275243((E)-3-(1-Cinnamyl-1H-1,2,3-triazol-4-yl)-N-hydroxy...)
Affinity DataIC50: 104nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts using Ac-Arg-Gly-Lys(Ac)-AMC substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50485175(CHEMBL2036471)
Affinity DataIC50: 105nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts using Ac-Arg-Gly-Lys(Ac)-AMC substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50485170(CHEMBL2036480)
Affinity DataIC50: 140nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts using Ac-Arg-Gly-Lys(Ac)-AMC substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50485166(CHEMBL2036472)
Affinity DataIC50: 178nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts using Ac-Arg-Gly-Lys(Ac)-AMC substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50485169(CHEMBL2036477)
Affinity DataIC50: 219nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts using Ac-Arg-Gly-Lys(Ac)-AMC substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50485171(CHEMBL2036481)
Affinity DataIC50: 333nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts using Ac-Arg-Gly-Lys(Ac)-AMC substrate by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed